GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC15A1 |
Alanine glutamate |
320000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Valacyclovir |
NA|4080000|740000|490000 |
431000|1420000|400000|1100000|3400000|NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC15A1 |
Aminolevulinic Acid |
790000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC15A1 |
beta-Alanylglycine |
7300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
5-Aminovaleric acid |
17400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
2-Amino-N-cyclohexylpropanamide |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
beta-alanyl-L-alanine |
4800000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Glycine, N-L-arginyl- |
NA |
NA|390000 |
NA |
270000|NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
H-Glu-Phe-Tyr-OH |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
(2R)-1-[(2S)-2,6-diaminohexanoyl]pyrrolidine-2-carboxylic acid |
NA|350000 |
NA|390000 |
NA |
190000|NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
H-Phe-Ser(Bz)-Chg-OH.TFA |
245470891.6 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
(2S)-2-[[(2S,5S)-5-amino-2-(benzoyloxymethyl)-4-oxo-6-phenylhexanoyl]amino]propanoic acid;2,2,2-trifluoroacetic acid |
323593656.9 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
(2S)-2-[[(2S,5S)-5-amino-2-(benzoyloxymethyl)-4-oxo-6-phenylhexanoyl]amino]pentanoic acid;2,2,2-trifluoroacetic acid |
251188643.2 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
(2S)-2-[[(2S,5S)-5-amino-2-(benzoyloxymethyl)-4-oxo-6-phenylhexanoyl]amino]-2-cyclohexylacetic acid;2,2,2-trifluoroacetic acid |
46773514.13 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
H-Phe-Ser(Bz)-Nva-OH.TFA |
123026877.1 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
H-Ala-Beta-Ala-OH |
4800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Methyl 4-(2-aminopropanoylamino)benzoate |
1100000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Lys-Arg |
NA |
7200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Prolylarginine |
2500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Aspartylglycine |
NA |
NA|810000 |
NA |
440000|NA |
NA |
NA |
BindingDB|TTD |