GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC12A5 |
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]benzamide |
NA |
NA |
NA |
544000 |
NA |
NA |
BindingDB |
SLC12A5 |
5-[(4-fluorobenzyl)thio]-2-methyl-4-nitro-1H-imidazole |
NA |
NA |
NA |
878000 |
NA |
NA |
BindingDB |
SLC12A5 |
1-Phenyl-3-(1-propylbenzimidazol-2-yl)thiourea |
NA |
NA |
NA |
60400000 |
NA |
NA |
BindingDB |
SLC12A5 |
3-[(6-Ethoxy-1,3-benzothiazol-2-yl)thio]-1-(3-methoxyphenyl)pyrrolidine-2,5-quinone |
NA |
NA |
NA |
244000 |
NA |
NA |
BindingDB |
SLC12A5 |
(6E)-6-[[2-(1,3-benzoxazol-2-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one |
NA |
NA |
NA |
367000|3040000 |
NA |
NA |
BindingDB |
SLC12A5 |
2-[3-Nitro-4-[[1-(phenylmethyl)-4-piperidinyl]amino]phenyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione |
NA |
NA |
NA |
221000 |
NA |
NA |
BindingDB |
SLC12A5 |
2-chloranyl-N-[3-(dimethylsulfamoyl)phenyl]-5,5-bis(oxidanylidene)-8,9,10,11-tetrahydro-7H-azepino[2,1-c][1,2,4]benzothiadiazine-3-carboxamide |
NA |
NA |
NA |
281000 |
NA |
NA |
BindingDB |
SLC12A5 |
N-(1-benzylpropyl)-2-[(2,4-diketo-1,3-dimethyl-quinazolin-6-yl)sulfonyl-methyl-amino]acetamide |
NA |
NA |
NA |
2410000 |
NA |
NA |
BindingDB |
SLC12A5 |
2-(2-naphthoxy)-N-(2-pyridylmethyleneamino)acetamide |
NA |
NA |
NA |
330000 |
NA |
NA |
BindingDB |
SLC12A5 |
1-(2-Chlorophenyl)-3-[(2-chlorophenyl)methyl]thiourea |
NA |
NA |
NA |
204000 |
NA |
NA |
BindingDB |
SLC13A3 |
Succinic Acid |
NA |
107000|NA |
NA |
NA|107000 |
NA |
NA |
PubChem |
SLC15A1 |
3-(4-Aminobutyl)-6-methylpiperazine-2,5-dione |
5400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Histidylglycine |
NA |
NA|340000 |
NA |
280000|NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Histidylalanine |
480000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
H-Trp-Gly-Tyr-OH |
240000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
(2S)-3-hydroxy-2-[[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid |
NA|2500000 |
1760000|5180000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
H-Ala-Phe-Pro-OH |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
(2S,3S,4R,5R)-2-(2-bromo-5,6-dichloro-benzimidazol-1-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol |
NA |
447000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Val-Val |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
SLC15A1 |
1-L-Alanyl-D-proline |
15000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |