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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC12A5 N-[(4-phenyl-1,3-thiazol-2-yl)methyl]benzamide NA NA NA 544000 NA NA BindingDB
SLC12A5 5-[(4-fluorobenzyl)thio]-2-methyl-4-nitro-1H-imidazole NA NA NA 878000 NA NA BindingDB
SLC12A5 1-Phenyl-3-(1-propylbenzimidazol-2-yl)thiourea NA NA NA 60400000 NA NA BindingDB
SLC12A5 3-[(6-Ethoxy-1,3-benzothiazol-2-yl)thio]-1-(3-methoxyphenyl)pyrrolidine-2,5-quinone NA NA NA 244000 NA NA BindingDB
SLC12A5 (6E)-6-[[2-(1,3-benzoxazol-2-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one NA NA NA 367000|3040000 NA NA BindingDB
SLC12A5 2-[3-Nitro-4-[[1-(phenylmethyl)-4-piperidinyl]amino]phenyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione NA NA NA 221000 NA NA BindingDB
SLC12A5 2-chloranyl-N-[3-(dimethylsulfamoyl)phenyl]-5,5-bis(oxidanylidene)-8,9,10,11-tetrahydro-7H-azepino[2,1-c][1,2,4]benzothiadiazine-3-carboxamide NA NA NA 281000 NA NA BindingDB
SLC12A5 N-(1-benzylpropyl)-2-[(2,4-diketo-1,3-dimethyl-quinazolin-6-yl)sulfonyl-methyl-amino]acetamide NA NA NA 2410000 NA NA BindingDB
SLC12A5 2-(2-naphthoxy)-N-(2-pyridylmethyleneamino)acetamide NA NA NA 330000 NA NA BindingDB
SLC12A5 1-(2-Chlorophenyl)-3-[(2-chlorophenyl)methyl]thiourea NA NA NA 204000 NA NA BindingDB
SLC13A3 Succinic Acid NA 107000|NA NA NA|107000 NA NA PubChem
SLC15A1 3-(4-Aminobutyl)-6-methylpiperazine-2,5-dione 5400000 NA NA NA NA NA TTD
SLC15A1 Histidylglycine NA NA|340000 NA 280000|NA NA NA BindingDB|TTD
SLC15A1 Histidylalanine 480000 NA NA NA NA NA TTD
SLC15A1 H-Trp-Gly-Tyr-OH 240000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (2S)-3-hydroxy-2-[[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid NA|2500000 1760000|5180000|NA NA NA NA NA BindingDB|TTD
SLC15A1 H-Ala-Phe-Pro-OH 110000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (2S,3S,4R,5R)-2-(2-bromo-5,6-dichloro-benzimidazol-1-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol NA 447000 NA NA NA NA BindingDB|TTD
SLC15A1 Val-Val NA 210000 NA NA NA NA BindingDB|PubChem
SLC15A1 1-L-Alanyl-D-proline 15000000 NA NA NA NA NA BindingDB|TTD