| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC12A5 |
1-(2,3-dihydroindol-1-yl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)-2-imidazol-1-ylbutane-1,4-dione |
NA |
NA |
NA |
113000|1770000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-(2-chloro-5-piperidin-1-ylsulfonylphenyl)-2-[(4-fluorophenyl)sulfonylamino]benzamide |
NA |
NA |
NA |
101000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-cyclohexyl-3-(furan-2-yl)-4-phenylbutanamide |
NA |
NA |
NA |
212000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-[2-(4-Chloro-2-methylphenoxy)phenyl]-3-oxopropanenitrile |
NA |
NA |
NA |
233000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-(4-Ethoxyphenyl)-3-{[phenyl(phenylthio)acetyl]amino}propanoic acid |
NA |
NA |
NA |
4060000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1-[2,2-Dimethyl-3-(phenethylthiocarbamoylamino)propyl]-3-phenethyl-thiourea |
NA |
NA |
NA |
165000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-(4-methyl-3-morpholin-4-ylsulfonylphenyl)-4-phenylsulfanylbutanamide |
NA |
NA |
NA |
408000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfinyl]ethanone |
NA |
NA |
NA |
1410000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-benzyl-2-[[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfonyl]acetamide |
NA |
NA |
NA |
110000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[2-(2-phenyl-1,3-thiazol-4-yl)ethyl]thiophene-2-carboxamide |
NA |
NA |
NA |
174000 |
NA |
NA |
BindingDB |
| SLC12A5 |
|
NA |
NA |
NA |
10100000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1-Benzyl-4-({2-[4-(benzyloxy)benzylidene]hydrazino}carbonyl)pyridinium chloride |
NA |
NA |
NA |
563000 |
NA |
NA |
BindingDB |
| SLC12A5 |
5-(4-chlorophenyl)-4-{[(E)-(5-methylthiophen-2-yl)methylidene]amino}-4H-1,2,4-triazole-3-thiol |
NA |
NA |
NA |
188000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(2Z)-1-cyclobutyl-2-(3-methyl-1,3-benzothiazol-2-ylidene)ethanone |
NA |
NA |
NA |
170000 |
NA |
NA |
BindingDB |
| SLC12A5 |
5-[2-(Benzyloxy)benzylidene]-3-methyl-2-thioxo-4-imidazolidinone |
NA |
NA |
NA |
1640000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[1-(5-bromo-2-thienyl)ethylideneamino]-piperonylamide |
NA |
NA |
NA |
726000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-hydroxy-N-[(5Z)-5-[(1-methylpyrrol-2-yl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzamide |
NA |
NA |
NA |
150000|385000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-({2-[(E)-(3-isopropyl-2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]phenoxy}methyl)benzoic acid |
NA |
NA |
NA |
218000 |
NA |
NA |
BindingDB |
| SLC12A5 |
|
NA |
NA |
NA |
145000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(E)-4-(1,3-benzothiazol-2-yl)-5-(2-nitrophenyl)pent-4-enoic acid |
NA |
NA |
NA |
350000|500000 |
NA |
NA |
BindingDB |