| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC12A5 |
|
NA |
NA |
NA |
233000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-methyl-N-{2-[(4-methylbenzyl)thio]ethyl}benzamide |
NA |
NA |
NA |
2690000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-[(1-bromo-2-naphthyl)oxy]-N-4H-1,2,4-triazol-4-ylacetamide |
NA |
NA |
NA |
459000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[(3-bromoanilino)-sulfanylidenemethyl]-3-phenylpropanamide |
NA |
NA |
NA |
296000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-chloro-N-[[4-(3-nitrophenyl)-1,3-thiazol-2-yl]carbamothioyl]benzamide |
NA |
NA |
NA |
139000|244000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-Phenyl-7-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one |
NA |
NA |
NA |
4610000 |
NA |
NA |
BindingDB |
| SLC12A5 |
7-[[5-(4-Methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one |
NA |
NA |
NA |
8870000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-(N-benzyl2,6-dichlorobenzenesulfonamido)propanoic acid |
NA |
NA |
NA |
86000000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(2E)-3-(1-benzyl-3-phenyl-1H-pyrazol-4-yl)prop-2-enoic acid |
NA |
NA |
NA |
13700000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[4-(dimethylsulfamoyl)phenyl]-2-quinazolin-4-ylsulfanylacetamide |
NA |
NA |
NA |
87700000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1-(4-chlorophenyl)-N-[2-[(4-fluorophenyl)methylsulfanyl]ethyl]-5-methylpyrazole-4-carboxamide |
NA |
NA |
NA |
471000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-[[5-(3,4-Dichlorophenyl)furan-2-yl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-one |
NA |
NA |
NA |
130000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-(Benzylamino)-5-nitrobenzoic acid |
NA |
NA |
NA |
1490000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-(4-morpholinyl)-3-nitro-N-[4-(4-pyridinylmethyl)phenyl]benzamide |
NA |
NA |
NA |
101000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-(1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl)-N-(3-methyl-1,3-benzothiazol-2-ylidene)propanamide |
NA |
NA |
NA |
120000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[2-(cyclopentylamino)-1-(4-ethoxyphenyl)-2-oxoethyl]-N-(3-hydroxypropyl)-5-phenyl-1H-pyrrole-2-carboxamide |
NA |
NA |
NA |
843000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-{2-[3,5-Dioxo-4-(2-phenylethyl)piperazin-1-YL]-2-oxoethyl}-N-methyl-2,1,3-benzothiadiazole-4-sulfonamide |
NA |
NA |
NA |
2270000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-{2-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}isoquinolin-1(2H)-one |
NA |
NA |
NA |
260000 |
NA |
NA |
BindingDB |
| SLC12A5 |
Ethyl 2-[(4-methoxy-1,3-benzothiazol-2-yl)amino]-4-methyl-1,3-thiazole-5-carboxylate |
NA |
NA |
NA |
155000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-({3-[(4-Benzylpiperidin-1-yl)carbonyl]piperidin-1-yl}sulfonyl)-2,1,3-benzoxadiazole |
NA |
NA |
NA |
1460000|3810000 |
NA |
NA |
BindingDB |