| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC12A5 |
3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-thienylsulfonyl)-4-piperidyl]methanone |
NA |
NA |
NA |
2650000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-(3-isopropoxypropyl)-2-[(2E)-2-(4-methylbenzylidene)-3-oxo-2,3-dihydro-4H-1,4-benzothiazin-4-yl]acetamide |
NA |
NA |
NA |
276000|964000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(2E)-2-[[4-methoxy-3-(morpholin-4-ylmethyl)phenyl]methylidene]-3,4-dihydronaphthalen-1-one |
NA |
NA |
NA |
219000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-({[4-(isobutyrylamino)-3-methoxyphenyl]amino}carbonothioyl)-2-furamide |
NA |
NA |
NA |
179675456 |
NA |
NA |
BindingDB |
| SLC12A5 |
5-[(2,5-dichlorophenoxy)methyl]-N-pyridin-3-ylfuran-2-carboxamide |
NA |
NA |
NA |
106000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-Methoxy-4-(4-morpholinylcarbonothioyl)phenyl (4-fluorophenyl)acetate |
NA |
NA |
NA |
137000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2',3'-Dihydroxy-4',6'-dimethoxychalcone |
NA |
NA |
NA |
486000 |
NA |
NA |
BindingDB |
| SLC12A5 |
Ethyl 4-[2-(tert-butylamino)-2-oxoethyl]-1-(4-fluorophenyl)pyrrolo[3,2-b]pyrrole-5-carboxylate |
NA |
NA |
NA |
51100000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-N'-[(2-methylphenoxy)acetyl]propanehydrazide |
NA |
NA |
NA |
432000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1-[(1-{6-[Benzyl(methyl)amino][1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperidin-3-yl)methyl]pyrrolidin-2-one |
NA |
NA |
NA |
9050000 |
NA |
NA |
BindingDB |
| SLC12A5 |
|
NA |
NA |
NA |
976000 |
NA |
NA |
BindingDB |
| SLC12A5 |
|
NA |
NA |
NA |
334000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N'-[2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetyl]-2-(4-ethylphenoxy)acetohydrazide |
NA |
NA |
NA |
1070000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-[2-({3-[2-(3,4-dihydro-2(1H)-isoquinolinyl)-2-oxoethyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene}methyl)phenoxy]acetamide |
NA |
NA |
NA |
10800000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[[(2-hydroxybenzoyl)amino]carbamothioyl]furan-2-carboxamide |
NA |
NA |
NA |
303000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(E)-N-[4-(2-methoxyphenyl)piperazine-1-carbothioyl]-3-phenylprop-2-enamide |
NA |
NA |
NA |
109000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-(5-methyl-1,2-oxazol-3-yl)-2-[3-[(4-methylphenyl)methyl]-4-oxoquinazolin-2-yl]sulfanylacetamide |
NA |
NA |
NA |
138000 |
NA |
NA |
BindingDB |
| SLC12A5 |
4-chloro-N-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]benzenesulfonamide |
NA |
NA |
NA |
112000|3290000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[2-(1H-indol-3-yl)ethyl]-2-morpholin-4-yl-5-piperidin-1-ylsulfonylbenzamide |
NA |
NA |
NA |
208000 |
NA |
NA |
BindingDB |
| SLC12A5 |
5-[(2,4-dichlorophenoxy)methyl]-N-(pyridin-3-ylmethyl)furan-2-carboxamide |
NA |
NA |
NA |
668000|2060000 |
NA |
NA |
BindingDB |