| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC12A5 |
(E)-3-(3-fluorophenyl)-1-(2-methyl-2,3-dihydroindol-1-yl)prop-2-en-1-one |
NA |
NA |
NA |
129000|192000 |
NA |
NA |
BindingDB |
| SLC12A5 |
|
NA |
NA |
NA |
41100000 |
NA |
NA |
BindingDB |
| SLC12A5 |
6-Methyl-3-({phenethyl-[1-(tetrahydro-furan-2-ylmethyl)-1H-tetrazol-5-ylmethyl]-amino}-methyl)-1H-quinolin-2-one |
NA |
NA |
NA |
244000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-[6-(4-Fluoro-phenyl)-pyridazin-3-ylsulfanyl]-1-(2-methyl-piperidin-1-yl)-ethanone |
NA |
NA |
NA |
8190000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-(1-Methyl-1H-benzoimidazol-2-ylmethylsulfanyl)-benzothiazole |
NA |
NA |
NA |
439000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[2-(2-Fluoro-phenyl)-ethyl]-3-(morpholine-4-sulfonyl)-benzenesulfonamide |
NA |
NA |
NA |
4040000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-{2-[4-(2-Fluoro-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-7-phenyl-3,7-dihydro-pyrazolo[3,4-d][1,2,3]triazin-4-one |
NA |
NA |
NA |
147000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-[1-(2,5-Dimethoxy-phenyl)-1H-tetrazol-5-ylsulfanyl]-N-phenethyl-acetamide |
NA |
NA |
NA |
233000|242000 |
NA |
NA |
BindingDB |
| SLC12A5 |
N-[1-(2-methoxyphenyl)-5-benzimidazolyl]benzenesulfonamide |
NA |
NA |
NA |
101000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1-(3,4-Dihydro-2H-quinolin-1-yl)-2-(5-phenylaminomethyl-[1,3,4]oxadiazol-2-ylsulfanyl)-ethanone |
NA |
NA |
NA |
1730000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(E)-4-(1,3-benzothiazol-2-yl)-5-(4-morpholin-4-yl-3-nitrophenyl)pent-4-enoic acid |
NA |
NA |
NA |
82100000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(E)-4-(1,3-benzothiazol-2-yl)-5-(3-nitro-4-pyrrolidin-1-ylphenyl)pent-4-enoic acid |
NA |
NA |
NA |
233000|290000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-(4-Chloro-phenyl)-4-{2-[4-(2-fluoro-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-4H-[1,2,4]oxadiazol-5-one |
NA |
NA |
NA |
228000 |
NA |
NA |
BindingDB |
| SLC12A5 |
Diacylglycerol Kinase Inhibitor Ii |
NA |
NA |
NA |
181000 |
NA |
NA |
BindingDB |
| SLC12A5 |
(4-Methoxyphenyl)(3-phenylpiperidin-1-yl)methanone |
NA |
NA |
NA |
110000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-(4,5-dihydro-1,3-thiazol-2-ylsulfanyl)-N-(4-phenyl-1,3-thiazol-2-yl)acetamide |
NA |
NA |
NA |
1890000 |
NA |
NA |
BindingDB |
| SLC12A5 |
2-[(2-Chlorophenyl)methylthio]-1-methylbenzimidazole |
NA |
NA |
NA |
260000 |
NA |
NA |
BindingDB |
| SLC12A5 |
|
NA |
NA |
NA |
144000 |
NA |
NA |
BindingDB |
| SLC12A5 |
3-(4-chlorophenyl)-4-[(E)-[(E)-3-(2-nitrophenyl)prop-2-enylidene]amino]-1H-1,2,4-triazole-5-thione |
NA |
NA |
NA |
148000 |
NA |
NA |
BindingDB |
| SLC12A5 |
1,3,4-Thiadiazole-2(3H)-thione, 5-anilino- |
NA |
NA |
NA |
633000 |
NA |
NA |
BindingDB |