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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC15A1 1-(2-Ammonio-3-phenylpropanoyl)pyrrolidine-2-carboxylate 130000 NA NA NA NA NA BindingDB
SLC15A1 1-[2-Ammonio-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carboxylate 160000 NA NA NA NA NA BindingDB
SLC15A1 2-{[2-ammonio-3-(1H-indol-2-yl)propanoyl]amino}propanoate 160000 NA NA NA NA NA BindingDB
SLC15A1 [(2-Ammoniopropanoyl)(methyl)amino]acetate 250000 NA NA NA NA NA BindingDB
SLC15A1 2-[(Ammonioacetyl)amino]-4-methylpentanoate 160000 NA NA NA NA NA BindingDB
SLC15A1 1-(2-Ammoniohexanoyl)pyrrolidine-2-carboxylate 160000 NA NA NA NA NA BindingDB
SLC15A1 1-(1,1''-Biphenyl-3-ylamino)-1-oxopropan-2-aminium 290000 NA NA NA NA NA BindingDB
SLC15A1 4-Ammonio-5-[(1-methyl-2-oxido-2-oxoethyl)amino]-5-oxopentanoate 250000 NA NA NA NA NA BindingDB
SLC15A1 [(2-Ammonio-3-phenylpropanoyl)(methyl)amino]acetate 210000 NA NA NA NA NA BindingDB
SLC15A1 2-[(2-Ammoniopropanoyl)amino]-2-methylpropanoate 1200000 NA NA NA NA NA BindingDB
SLC15A1 1-{[4-(Methoxycarbonyl)phenyl]amino}-1-oxopropan-2-aminium 1100000 NA NA NA NA NA BindingDB
SLC15A1 2-[(R)-2-((S)-2-Amino-propionylamino)-3-phenyl-propionylamino]-propionic acid 19000000 NA NA NA NA NA BindingDB
SLC15A1 Val-Ala-Leu 140000 NA NA NA NA NA BindingDB|TTD
SLC15A1 2-((R)-2-Amino-3-phenyl-propionylamino)-propionic acid 7000000|7100000 NA NA NA NA NA BindingDB
SLC15A1 7-((S)-2-Azido-2-phenyl-acetylamino)-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid anion 15000000 NA NA NA NA NA BindingDB
SLC15A1 7-[[(2S)-2-azido-2-phenylacetyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 15000000 NA NA NA NA NA TTD
SLC15A1 Cyclohexanecarboxylic acid ((S)-2-amino-propionyl)-amide 1500000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (S)-2-({(S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carbonyl}-amino)-3-methyl-pentanoic acid 250000 NA NA NA NA NA BindingDB
SLC15A1 (S)-3-Amino-N-((S)-1-carbamoyl-ethyl)-succinamic acid 5400000 NA NA NA NA NA BindingDB|TTD
SLC15A1 ((S)-2-Amino-propionyl)-(3-fluoro-phenyl)-carbamic acid 3100000 NA NA NA NA NA BindingDB|TTD