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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC15A1 H-Trp-Trp-Trp-OH 170000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (S)-2-[(S)-2-(2-Amino-4-methylsulfanyl-butyrylamino)-4-methylsulfanyl-butyrylamino]-4-methylsulfanyl-butyric acid 520000 NA NA NA NA NA BindingDB
SLC15A1 (S)-3-((S)-2,6-Diamino-hexanoylamino)-4-oxo-butyric acid 330000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (S)-2-{(2S,3R)-2-[((S)-2-Amino-4-methyl-pentanoyl)-methyl-amino]-3-hydroxy-butyrylamino}-4-methyl-pentanoic acid 110000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (S)-2-[(S)-2-(2-Amino-propionylamino)-propionylamino]-propionic acid 7900000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (S)-2-[(S)-2-Amino-3-(4-phenoxy-phenyl)-propionylamino]-propionic acid 1400000 NA NA NA NA NA BindingDB|TTD
SLC15A1 (R)-6-Amino-2-((R)-2-amino-propionylamino)-hexanoic acid 30000000 NA NA NA NA NA TTD
SLC15A1 ((S)-2-Amino-propionyl)-phenyl-carbamic acid 2900000 NA NA NA NA NA BindingDB|TTD
SLC15A1 [2-(7-{2-(2-Amino-thiazol-4-yl)-2-[(Z)-methoxyimino]-acetylamino}-2-carboxy-8-oxo-5-thia-1-aza-bicyclo[4.2.0]oct-2-en-3-ylmethylsulfanyl)-5-methyl-thiazol-4-yl]-acetic acid anion 22000000 NA NA NA NA NA BindingDB
SLC15A1 Phe-Leu-Leu 140000 NA NA NA NA NA BindingDB|TTD
SLC15A1 Pro-Leu NA NA|620000 NA 250000|NA NA NA BindingDB|TTD
SLC15A1 Ac-Phe-di-iodo-Tyr NA 230000 NA NA NA NA BindingDB|TTD
SLC15A1 1-Oxo-1-piperidin-1-ylpropan-2-aminium 12900000 NA NA NA NA NA BindingDB
SLC15A1 L-Valine[3-[(Aminoiminomethyl)amino]phenyl]methyl Ester NA 650000 NA NA NA NA BindingDB|TTD
SLC15A1 L-Isoleucine[3-[(Aminoiminomethyl)amino]phenyl]methyl Ester NA 630000 NA NA NA NA BindingDB|TTD
SLC15A1 L-Phenylalanine[3-[(Aminoiminomethyl)amino]phenyl]methyl Ester NA 2330000 NA NA NA NA BindingDB|TTD
SLC15A1 (2S)-2-{[(2S)-2-aminohexanoyl]amino}propanoic acid 140000 NA NA NA NA NA TTD
SLC15A1 Cefamandole 8100000 NA NA NA NA NA BindingDB|PubChem|TTD
SLC15A1 (S)-2-amino-3-methylbutanoic benzoic anhydride NA 390000 NA NA NA NA BindingDB|TTD
SLC15A1 (2S,3S)-2-amino-3-methylpentanoic benzoic anhydride NA 630000 NA NA NA NA BindingDB|TTD