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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC1A1 DL-Tboa NA 161000 NA NA NA NA BindingDB
SLC1A1 4-{[(5Z)-3-(2-Ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}benzoic acid NA 300000 NA NA NA NA TTD
SLC1A1 Cysteine NA 161000|NA NA NA|161000 NA NA PubChem
SLC1A1 Ethyl (5-{[5-(4-morpholinyl)-2-furyl]methylene}-2,4-dioxo-1,3-thiazolidin-3-yl)acetate NA 300000 NA NA NA NA TTD
SLC1A1 3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]-4-methylbenzoic acid NA 300000 NA NA NA NA TTD
SLC1A1 (4r)-4-{3-[hydroxy(Methyl)amino]-3-Oxopropyl}-L-Glutamic Acid NA 3000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-[3-oxo-3-(prop-2-ynylamino)propyl]pentanedioic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-(3-anilino-3-oxopropyl)pentanedioic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-[3-(diethylamino)-3-oxopropyl]pentanedioic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-(3-oxo-3-piperidin-1-ylpropyl)pentanedioic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-[3-oxo-3-(phenylmethoxyamino)propyl]pentanedioic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-(2-cyanoethyl)pentanedioic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-[3-(hydroxyamino)-3-oxopropyl]pentanedioic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-(2-aminoethyl)pentanedioic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-2-amino-4-(3-aminopropyl)pentanedioic acid NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-azepane-2,4-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A1 (2S,4R)-4-(4-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride NA 1000000 NA NA NA NA TTD
SLC1A1 (2S,4R)-4-(3-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride NA 1000000 NA NA NA NA TTD
SLC1A2 2-Amino-3-(3-hydroxy-5-methyl-3H-[1,2,3]triazol-4-yl)-propionic acid NA 490000 NA NA NA NA TTD
SLC1A2 (3S,5S)-2-aza-bicyclo[2.2.1]heptane-3,5-dicarboxylic acid 400000 NA NA NA NA NA TTD