GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC1A2 |
(RS)-2-amino-3-(1-hydroxy-1,2,3-triazol-5-yl)propionate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(1-hydroxy-5-methyl-1H-imidazol-2-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(2-hydroxy-4-methyl-2H-pyrazol-3-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic acid |
NA |
430000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(3-hydroxy-2-methyl-3H-imidazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(3-hydroxy-5-methyl-3H-imidazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC1A2 |
(1R,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(1S,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(1R,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(1S,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
2-Amino-3-(2,5-dihydro-5-oxo-4-isoxazolyl)propanoic acid |
NA |
240000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S,3R)-2-amino-3-(benzenesulfonamido)butanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S)-2-amino-3-(phenoxycarbonylamino)butanedioic acid |
NA |
316227.77 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S)-2-amino-3-(4-phenyltriazol-1-yl)butanedioic acid |
NA |
501187.23 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S)-2-amino-3-[(3-carboxyphenyl)sulfonylamino]butanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S)-2-amino-3-[benzenesulfonyl(methyl)amino]butanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S)-2-amino-3-[(4-methylsulfonylphenyl)sulfonylamino]butanedioic acid |
NA |
316227.77 |
NA |
NA |
NA |
NA |
TTD |