| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC1A2 |
4-chloro-3-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-chloro-3-[5-[(Z)-(3-methyl-2,4-dioxo-thiazolidin-5-ylidene)methyl]-2-furyl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
Ethyl (5-{[5-(2-bromo-4-methylphenyl)-2-furyl]methylene}-2,4-dioxo-1,3-thiazolidin-3-yl)acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-chloro-3-[5-[(Z)-[3-[2-(4-methylanilino)-2-oxo-ethyl]-2,4-dioxo-thiazolidin-5-ylidene]methyl]-2-furyl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-Thiazolidineacetic acid, 5-[[5-(5-carboxy-2-chlorophenyl)-2-furanyl]methylene]-2,4-dioxo-, methyl ester, (5Z)- |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl [(5Z)-5-{[5-(4-chloro-3-nitrophenyl)furan-2-yl]methylidene}-2,4-dioxo-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
2-chloro-5-(5-{(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}furan-2-yl)benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-5-[[5-(2-chloro-5-nitrophenyl)furan-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-2,4-dioxo-5-[(5-phenylfuran-2-yl)methylidene]-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-5-[(5-methylfuran-2-yl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-chloro-3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-5-[[5-(2,5-dichlorophenyl)furan-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-5-[[5-(2-chloro-4-nitrophenyl)furan-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-2,4-dioxo-5-[(5-phenylsulfanylfuran-2-yl)methylidene]-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl [(5Z)-2,4-dioxo-5-{[5-(piperidin-1-yl)furan-2-yl]methylidene}-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-4-(3-Amino-3-oxopropyl)glutamic acid |
290000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(4r)-4-[3-(Methylamino)-3-Oxopropyl]-L-Glutamic Acid |
630957.34 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-4-(3-Benzylamino-3-oxopropyl)glutamic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4S)-4-(Hydroxymethyl)glutamic Acid |
125892.54 |
NA |
NA |
NA |
NA |
NA |
TTD |