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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC1A2 (2S,4R)-4-(4-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride NA 1000000 NA NA NA NA TTD
SLC1A2 (2S,4R)-4-(3-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride NA 1000000 NA NA NA NA TTD
SLC1A3 (2S,1''S,2''R)-2-(2''-Carboxycyclobutyl)glycine 200000 NA NA NA NA NA BindingDB
SLC1A3 2-Amino-3-(3-hydroxy-5-methyl-3H-[1,2,3]triazol-4-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 (3S,5S)-2-aza-bicyclo[2.2.1]heptane-3,5-dicarboxylic acid 400000 NA NA NA NA NA TTD
SLC1A3 (2S,4R)-4-pentylglutamic acid 120000|117489.76 NA NA NA NA NA BindingDB|TTD
SLC1A3 Dihydrokainic acid NA 3000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(1-hydroxy-5-methyl-1H-imidazol-2-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(2-hydroxy-4-methyl-2H-pyrazol-3-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(3-hydroxy-2-methyl-3H-imidazol-4-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 2-Amino-3-(3-hydroxy-5-methyl-3H-imidazol-4-yl)-propionic acid NA 1000000 NA NA NA NA TTD
SLC1A3 (1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarboxylic acid 127000 NA NA NA NA NA BindingDB|TTD
SLC1A3 alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID NA 1000000 NA NA NA NA PubChem|TTD
SLC1A3 (1R,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A3 (1S,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A3 (1R,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD
SLC1A3 (1S,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid NA 300000 NA NA NA NA TTD