GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC1A2 |
(2S,4R)-4-(4-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A2 |
(2S,4R)-4-(3-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,1''S,2''R)-2-(2''-Carboxycyclobutyl)glycine |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
SLC1A3 |
2-Amino-3-(3-hydroxy-5-methyl-3H-[1,2,3]triazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(3S,5S)-2-aza-bicyclo[2.2.1]heptane-3,5-dicarboxylic acid |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-4-pentylglutamic acid |
120000|117489.76 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
Dihydrokainic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(1-hydroxy-5-methyl-1H-imidazol-2-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(2-hydroxy-4-methyl-2H-pyrazol-3-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(3-hydroxy-2-methyl-3H-imidazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(1-hydroxy-1H-imidazol-2-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(3-hydroxy-3H-imidazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-3-(3-hydroxy-5-methyl-3H-imidazol-4-yl)-propionic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarboxylic acid |
127000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
alpha-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC1A3 |
(1R,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(1S,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(1R,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(1S,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |