| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC1A3 |
2-Amino-3-(2,5-dihydro-5-oxo-4-isoxazolyl)propanoic acid |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC1A3 |
(2S,3R)-2-amino-3-(benzenesulfonamido)butanedioic acid |
NA |
199526|200000|199526.23 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC1A3 |
(2S)-2-amino-3-(phenoxycarbonylamino)butanedioic acid |
NA |
999000|1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| SLC1A3 |
(2S)-2-amino-3-[(4-tert-butylphenyl)sulfonylamino]butanedioic acid |
NA |
300000|316228 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC1A3 |
(2S)-2-amino-3-(4-phenyltriazol-1-yl)butanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
(2S)-2-amino-3-benzamidobutanedioic acid |
NA |
300000|316228 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC1A3 |
(2S)-2-amino-3-[(3-carboxyphenyl)sulfonylamino]butanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
(2S)-2-amino-3-[benzenesulfonyl(methyl)amino]butanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
(2S)-2-amino-3-[(4-methylsulfonylphenyl)sulfonylamino]butanedioic acid |
NA |
300000|316228 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC1A3 |
(2S,4R)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
(2S,4S)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
4-chloro-3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]thiophen-2-yl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
4-chloro-3-[4-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
4-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-3-hydroxybenzoic acid |
NA |
316227.77 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
3-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]propanoic acid |
NA |
316227.77 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-4-hydroxybenzoic acid |
NA |
316227.77 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-2-hydroxybenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
2-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
2-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-4-hydroxyphenyl]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A3 |
(E)-3-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]prop-2-enoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |