GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC1A3 |
(2S,4R)-4-(3-Propylamino-3-oxopropyl)glutamic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-4-(3-Benzylamino-3-oxopropyl)glutamic acid |
NA|1000000 |
1000000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acid |
NA|1000000 |
1000000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
(2S,4S)-4-(Hydroxymethyl)glutamic Acid |
NA|3000000 |
3000000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
(2S,4S)-4-(Benzyloxymethyl)glutamic Acid |
NA|450000 |
1000000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
(2S,4S)-4-(2-Hydroxy-2-oxoethyl)glutamic Acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2s,4r)-4-(3-Methoxy-3-Oxopropyl) Glutamic Acid |
NA|1000000 |
1000000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
(2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic Acid |
NA|3000000 |
3000000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
Glutamic Acid |
NA |
398000|NA |
NA |
NA|398000 |
NA |
NA |
PubChem |
SLC1A3 |
Hinokinin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(1s,2r)-2-[(S)-Amino(Carboxy)methyl]cyclobutanecarboxylic Acid |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
ethyl (1E)-N-(3-cyano-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydrochromen-2-yl)methanimidate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]benzoic acid |
NA |
316227.77 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
DL-Tboa |
NA |
637000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC1A3 |
4-{[(5Z)-3-(2-Ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
Cysteine |
NA |
376000|NA |
NA |
NA|376000 |
NA |
NA |
PubChem |
SLC1A3 |
Aspartic Acid |
NA |
NA|398000 |
NA |
398000|NA |
NA |
NA |
PubChem |
SLC1A3 |
Ethyl (5-{[5-(4-morpholinyl)-2-furyl]methylene}-2,4-dioxo-1,3-thiazolidin-3-yl)acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-Amino-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydropyrano[3,2-c]pyridine-3-carbonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
2-amino-5-oxo-4,7-diphenyl-7,8-dihydro-4H-pyrano[3,2-c]pyran-3-carbonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |