GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC1A3 |
(4r)-4-{3-[hydroxy(Methyl)amino]-3-Oxopropyl}-L-Glutamic Acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-[3-oxo-3-(prop-2-ynylamino)propyl]pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-(3-anilino-3-oxopropyl)pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-[3-(diethylamino)-3-oxopropyl]pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-(3-oxo-3-piperidin-1-ylpropyl)pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-[3-oxo-3-(phenylmethoxyamino)propyl]pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-(2-cyanoethyl)pentanedioic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC1A3 |
(2S,4R)-2-amino-4-[3-(hydroxyamino)-3-oxopropyl]pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-(2-aminoethyl)pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-2-amino-4-(3-aminopropyl)pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-azepane-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(1R,2S)-2-[(S)-amino(carboxy)methyl]-2-methylcyclobutane-1-carboxylic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
D-Aspartic Acid |
NA |
NA|398000 |
NA |
398000|NA |
NA |
NA |
PubChem |
SLC1A3 |
(2S,4R)-4-(4-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A3 |
(2S,4R)-4-(3-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC1A4 |
Proline |
NA |
2139000 |
NA |
NA |
NA |
NA |
PubChem |
SLC1A4 |
Hydroxyproline |
NA |
188000|2000000 |
NA |
NA |
NA |
NA |
PubChem |
SLC1A4 |
Serine |
NA |
292000 |
NA |
NA |
NA |
NA |
PubChem |
SLC1A4 |
Glutamine |
NA |
3373000 |
NA |
NA |
NA |
NA |
PubChem |
SLC1A4 |
Asparagine |
NA |
656000 |
NA |
NA |
NA |
NA |
PubChem |