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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SLC1A4
D-Serine
NA
3937000
NA
NA
NA
NA
PubChem
SLC1A5
(2S)-2-amino-5-(2-morpholin-4-ylanilino)-5-oxopentanoic acid
NA
664000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-5-[2-(1,3-benzothiazol-2-yl)anilino]-5-oxopentanoic acid
NA
436000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-5-[2-(morpholin-4-ylmethyl)anilino]-5-oxopentanoic acid
NA
312000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-5-oxo-5-(2-piperidin-1-ylanilino)pentanoic acid
NA
776000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-5-oxo-5-[2-(2-pyridin-4-ylethyl)anilino]pentanoic acid
NA
832000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-5-[[2-(morpholin-4-ylsulfonylmethyl)phenyl]methylamino]-5-oxopentanoic acid
NA
677000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-5-[[2-[(4-methylpiperazin-1-yl)methyl]phenyl]methylamino]-5-oxopentanoic acid
NA
697000
NA
NA
NA
NA
TTD
SLC1A5
(2S)-2-amino-4-[bis[[2-(4-fluorophenoxy)phenyl]methyl]amino]butanoic acid
NA
141700
NA
NA
NA
NA
TTD
SLC1A5
Proline
NA
10000000
NA
NA
NA
NA
PubChem
SLC1A5
S-Benzylcysteine
780000
NA
NA
NA
NA
NA
GtoPDB
SLC1A5
Hydroxyproline
NA
3475000|2000000
NA
NA
NA
NA
PubChem
SLC1A5
Serine
NA
822000
NA
NA
NA
NA
PubChem
SLC1A5
Glutamine
NA
541000
NA
NA
NA
NA
PubChem
SLC1A5
Asparagine
NA
674000
NA
NA
NA
NA
PubChem
SLC1A5
D-Serine
NA
4913000
NA
NA
NA
NA
PubChem
SLC1A5
O-benzyl-L-serine
900000
NA
NA
NA
NA
NA
GtoPDB
SLC1A5
N5-(4-Nitrophenyl)-L-glutamine
NA
1200000
NA
NA
NA
NA
TTD
SLC22A1
Thiamine
NA
4354000
NA
NA
NA
NA
BindingDB|PubChem
SLC22A1
Eltrombopag
103000
NA
NA
NA
NA
NA
PubChem
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