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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC1A4 D-Serine NA 3937000 NA NA NA NA PubChem
SLC1A5 (2S)-2-amino-5-(2-morpholin-4-ylanilino)-5-oxopentanoic acid NA 664000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-5-[2-(1,3-benzothiazol-2-yl)anilino]-5-oxopentanoic acid NA 436000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-5-[2-(morpholin-4-ylmethyl)anilino]-5-oxopentanoic acid NA 312000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-5-oxo-5-(2-piperidin-1-ylanilino)pentanoic acid NA 776000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-5-oxo-5-[2-(2-pyridin-4-ylethyl)anilino]pentanoic acid NA 832000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-5-[[2-(morpholin-4-ylsulfonylmethyl)phenyl]methylamino]-5-oxopentanoic acid NA 677000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-5-[[2-[(4-methylpiperazin-1-yl)methyl]phenyl]methylamino]-5-oxopentanoic acid NA 697000 NA NA NA NA TTD
SLC1A5 (2S)-2-amino-4-[bis[[2-(4-fluorophenoxy)phenyl]methyl]amino]butanoic acid NA 141700 NA NA NA NA TTD
SLC1A5 Proline NA 10000000 NA NA NA NA PubChem
SLC1A5 S-Benzylcysteine 780000 NA NA NA NA NA GtoPDB
SLC1A5 Hydroxyproline NA 3475000|2000000 NA NA NA NA PubChem
SLC1A5 Serine NA 822000 NA NA NA NA PubChem
SLC1A5 Glutamine NA 541000 NA NA NA NA PubChem
SLC1A5 Asparagine NA 674000 NA NA NA NA PubChem
SLC1A5 D-Serine NA 4913000 NA NA NA NA PubChem
SLC1A5 O-benzyl-L-serine 900000 NA NA NA NA NA GtoPDB
SLC1A5 N5-(4-Nitrophenyl)-L-glutamine NA 1200000 NA NA NA NA TTD
SLC22A1 Thiamine NA 4354000 NA NA NA NA BindingDB|PubChem
SLC22A1 Eltrombopag 103000 NA NA NA NA NA PubChem