Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
SLC22A1 | Methylnaltrexone | NA | 234000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A1 | Indinavir | NA | 208000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A1 | Tetraethylammonium | 158000|161000|163000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A1 | Noroxycodone | NA | 199820 | NA | NA | NA | NA | BindingDB |
SLC22A1 | Famotidine | NA | 300000 | NA | NA | NA | NA | PubChem |
SLC22A1 | Tetramethylammonium | 12400000 | NA | NA | NA | NA | NA | BindingDB |
SLC22A1 | N-Methylnicotinamide | 7700000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A1 | Tetrapropylammonium | 102000 | NA | NA | NA | NA | NA | BindingDB |
SLC22A11 | Indican | 181000|181300 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A11 | Octanoate | 235500 | NA | NA | NA | NA | NA | BindingDB |
SLC22A11 | Zonampanel | NA | 300000 | NA | NA | NA | NA | PubChem |
SLC22A11 | Cimetidine | NA | 2000000 | NA | NA | NA | NA | PubChem |
SLC22A11 | Octanoic Acid | 235500 | NA | NA | NA | NA | NA | PubChem |
SLC22A11 | Piroxicam | 107800 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A11 | Pravastatin | NA | 591000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A11 | CID 57049232 | 366400 | NA | NA | NA | NA | NA | BindingDB |
SLC22A11 | Betamipron | NA|502000 | 483000|NA | NA | NA | NA | NA | BindingDB |
SLC22A12 | Allopurinol | NA | 300000 | NA | NA | NA | NA | PubChem |
SLC22A12 | N-(4-(2H-tetrazol-5-yl)phenyl)-6-hydroxy-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | NA | 147000 | NA | NA | NA | NA | BindingDB |
SLC22A12 | [5-Bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanylmethanesulfonamide | NA | 365000 | NA | NA | NA | NA | TTD |