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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC22A12 2,6-Dibromo-4-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]phenol NA 119000 NA NA NA NA TTD
SLC22A2 2-Tert-butyl-4-[(2,4-diaminopyrimidin-5-yl)methyl]-6-methylphenol NA 4124120 NA NA NA NA BindingDB
SLC22A2 2-[4-[(2,4-Diaminopyrimidin-5-yl)methyl]-2,6-diethylphenoxy]ethanol NA 1267220 NA NA NA NA BindingDB
SLC22A2 Tetrabutylammonium NA 120000 NA NA NA NA BindingDB
SLC22A2 Zantac NA 1617000 NA NA NA NA BindingDB|PubChem
SLC22A2 Maraviroc NA 255000 NA NA NA NA BindingDB|PubChem
SLC22A2 Metformin NA 1700000 NA NA NA NA BindingDB|PubChem
SLC22A2 Mylanta AR 1800000 NA NA NA NA NA BindingDB
SLC22A2 Indinavir NA 142000 NA NA NA NA BindingDB|PubChem
SLC22A2 Tetraethylammonium NA 156000 NA NA NA NA BindingDB|PubChem
SLC22A2 Famotidine 1800000 NA NA NA NA NA PubChem
SLC22A2 Aripiprazole NA 239000 NA NA NA NA BindingDB|PubChem
SLC22A2 Tetramethylammonium NA|180000 150000|NA NA NA NA NA BindingDB
SLC22A2 N-Methylnicotinamide 266000 NA NA NA NA NA BindingDB|PubChem
SLC22A2 Metiprenaline 570000 NA NA NA NA NA BindingDB
SLC22A2 Tetrapropylammonium NA 128000 NA NA NA NA BindingDB
SLC22A3 N-(4-benzylphenyl)guanidine NA 452500 NA NA NA NA BindingDB|TTD
SLC22A3 Clonidine 373000 NA NA NA NA NA BindingDB|PubChem
SLC22A3 Guanidine NA|6201000 2200000|NA NA NA NA NA BindingDB|PubChem|TTD
SLC22A3 Ritonavir NA 300000 NA NA NA NA PubChem|TTD