Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
SLC22A3 | Nifekalant | NA | 146000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
SLC22A3 | Pantoprazole | NA | 137000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
SLC22A3 | Procainamide | 738000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A3 | Indinavir | NA | 500000 | NA | NA | NA | NA | PubChem|TTD |
SLC22A3 | Tetraethylammonium | NA|1372000 | 10300000|NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A3 | Histamine | 140000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A5 | Cefepime | NA | 1700000 | NA | NA | NA | NA | PubChem |
SLC22A5 | Cephaloridine | NA | 230000 | NA | NA | NA | NA | PubChem |
SLC22A6 | 2,2-Dimethylbutyric acid | NA | 3862000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A6 | Cyclic-hpmpc | NA | 1100000 | NA | NA | NA | NA | BindingDB |
SLC22A6 | (2S)-2-amino-3-[(Z)-1,2-dichloroethenyl]sulfanylpropanoic acid | NA | 208000 | NA | NA | NA | NA | BindingDB |
SLC22A6 | 3-[2-(6-aminopurin-9-yl)ethoxymethyl-[3-[(4R)-4-[(3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydroxy-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]pentanoyl]oxypropoxy]phosphoryl]oxypropyl (2R)-2-amino-4-methylpentanoate | NA | 285000 | NA | NA | NA | NA | BindingDB |
SLC22A6 | p-Aminohippuric acid | NA | 127000 | NA | NA | NA | NA | PubChem |
SLC22A6 | Cimetidine | NA | 492000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A6 | Salicylic Acid | NA | 280000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A6 | Cephradine | NA | 1600000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A6 | tert-butyl N-[(2S)-3-(1H-indol-3-yl)-1-oxo-1-[2-(2-oxo-1-phenylpyrrolidin-3-yl)sulfanylcarbonylhydrazinyl]propan-2-yl]carbamate | NA | 127000 | NA | NA | NA | NA | BindingDB |
SLC22A6 | Oseltamivir Acid | 45100000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A6 | Phenacetin | NA | 200000 | NA | NA | NA | NA | BindingDB|PubChem |
SLC22A6 | Pravastatin | NA | 408000 | NA | NA | NA | NA | BindingDB|PubChem |