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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC22A3 Nifekalant NA 146000 NA NA NA NA BindingDB|PubChem|TTD
SLC22A3 Pantoprazole NA 137000 NA NA NA NA BindingDB|PubChem|TTD
SLC22A3 Procainamide 738000 NA NA NA NA NA BindingDB|PubChem
SLC22A3 Indinavir NA 500000 NA NA NA NA PubChem|TTD
SLC22A3 Tetraethylammonium NA|1372000 10300000|NA NA NA NA NA BindingDB|PubChem
SLC22A3 Histamine 140000 NA NA NA NA NA BindingDB|PubChem
SLC22A5 Cefepime NA 1700000 NA NA NA NA PubChem
SLC22A5 Cephaloridine NA 230000 NA NA NA NA PubChem
SLC22A6 2,2-Dimethylbutyric acid NA 3862000 NA NA NA NA BindingDB|PubChem
SLC22A6 Cyclic-hpmpc NA 1100000 NA NA NA NA BindingDB
SLC22A6 (2S)-2-amino-3-[(Z)-1,2-dichloroethenyl]sulfanylpropanoic acid NA 208000 NA NA NA NA BindingDB
SLC22A6 3-[2-(6-aminopurin-9-yl)ethoxymethyl-[3-[(4R)-4-[(3R,5S,7S,8R,9S,10S,13R,14S,17R)-3,7-dihydroxy-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]pentanoyl]oxypropoxy]phosphoryl]oxypropyl (2R)-2-amino-4-methylpentanoate NA 285000 NA NA NA NA BindingDB
SLC22A6 p-Aminohippuric acid NA 127000 NA NA NA NA PubChem
SLC22A6 Cimetidine NA 492000 NA NA NA NA BindingDB|PubChem
SLC22A6 Salicylic Acid NA 280000 NA NA NA NA BindingDB|PubChem
SLC22A6 Cephradine NA 1600000 NA NA NA NA BindingDB|PubChem
SLC22A6 tert-butyl N-[(2S)-3-(1H-indol-3-yl)-1-oxo-1-[2-(2-oxo-1-phenylpyrrolidin-3-yl)sulfanylcarbonylhydrazinyl]propan-2-yl]carbamate NA 127000 NA NA NA NA BindingDB
SLC22A6 Oseltamivir Acid 45100000 NA NA NA NA NA BindingDB|PubChem
SLC22A6 Phenacetin NA 200000 NA NA NA NA BindingDB|PubChem
SLC22A6 Pravastatin NA 408000 NA NA NA NA BindingDB|PubChem