| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC1A2 |
(2S,4S)-4-(Benzyloxymethyl)glutamic Acid |
290000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4S)-4-(2-Hydroxy-2-oxoethyl)glutamic Acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2s,4r)-4-(3-Methoxy-3-Oxopropyl) Glutamic Acid |
158489.32 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-4-(3-Hydroxy-3-oxopropyl)glutamic Acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
2-Amino-4-(1,3-benzodioxol-5-yl)-5-oxo-7-phenyl-4,6,7,8-tetrahydrochromene-3-carbonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-{[(5Z)-3-(2-Ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
Ethyl (5-{[5-(4-morpholinyl)-2-furyl]methylene}-2,4-dioxo-1,3-thiazolidin-3-yl)acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]-4-methylbenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(4r)-4-{3-[hydroxy(Methyl)amino]-3-Oxopropyl}-L-Glutamic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-[3-oxo-3-(prop-2-ynylamino)propyl]pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-(3-anilino-3-oxopropyl)pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-[3-(diethylamino)-3-oxopropyl]pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-(3-oxo-3-piperidin-1-ylpropyl)pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-[3-oxo-3-(phenylmethoxyamino)propyl]pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-[2-(phenylmethoxycarbonylamino)ethyl]pentanedioic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-[3-(hydroxyamino)-3-oxopropyl]pentanedioic acid |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-(2-aminoethyl)pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-2-amino-4-(3-aminopropyl)pentanedioic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4R)-azepane-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |