| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC1A2 |
(2S,4R)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(2S,4S)-4-(2-carboxyphenoxy)pyrrolidine-2-carboxylic acid;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-chloro-3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]thiophen-2-yl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-chloro-3-[4-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]-4-methoxybenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-3-hydroxybenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]propanoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]naphthalene-2-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-4-hydroxybenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-2-hydroxybenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-chloro-3-[5-[(Z)-[3-(1-methoxy-1-oxopropan-2-yl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
2-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]-4-fluorobenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
2-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-4-hydroxyphenyl]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
(E)-3-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenyl]prop-2-enoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
ethyl 2-[(5Z)-2,4-dioxo-5-[[3-(2H-tetrazol-5-yl)phenyl]methylidene]-1,3-thiazolidin-3-yl]acetate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
4-Chloro-3-[5-[[3-(2-ethoxy-2-oxoethyl)-2,4-dioxoimidazolidin-1-yl]methyl]furan-2-yl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[3-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-4-hydroxyphenyl]propanoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]-4-phenylmethoxybenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SLC1A2 |
3-chloro-4-[5-[(Z)-[3-(2-ethoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]furan-2-yl]benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |