GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC47A1 |
Enalapril |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A1 |
Thiabendazole |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A1 |
Dexamethasone |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A1 |
Aripiprazole |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC47A1 |
Methylergonovine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A1 |
Nicotinic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A1 |
Azacitidine |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A2 |
Pimozide |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC47A2 |
Maraviroc |
NA |
297000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC47A2 |
(3H)granisetron |
NA |
311000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC47A2 |
Pantoprazole |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
SLC47A2 |
Rimantadine |
NA |
288000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC47A2 |
Risperidone |
NA |
291000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC47A2 |
Indinavir |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
SLC47A2 |
Aripiprazole |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
SLC5A1 |
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((3-hydroxypropoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol |
NA |
103000 |
NA |
NA |
NA |
NA |
TTD |
SLC5A1 |
(2S,3R,4R,5S,6R)-2-(4-chloro-2-((2,2-difluoropropoxy)methyl)-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
SLC5A1 |
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2,2,2-trifluoroethoxy)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
SLC5A1 |
Phlorizin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
SLC5A1 |
(Z)-1-[2,4-dihydroxy-6-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]-3-(4-hydroxyphenyl)prop-2-en-1-one |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |