| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A1 |
2,4-dichloro-N-(1-prop-2-ynylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
1-Benzyl-piperidin-4-yl benzoate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
N-(1-benzylpiperidin-4-yl)-2-methylpropanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
(3R,5R)-5-[2-[(2E)-2-[[5-[2-chloro-4-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]ethyl]piperidine-3-carboxylic acid |
NA |
134896|169824|169824.37 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
(3R,5S)-5-[[(2E)-2-[(5-naphthalen-1-ylfuran-2-yl)methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid |
NA |
169824 |
NA |
NA |
NA |
NA |
BindingDB |
| SLC6A1 |
(3R,5R)-5-[2-[(2E)-2-[[5-(2,4-dichlorophenyl)furan-2-yl]methylidene]hydrazinyl]ethyl]piperidine-3-carboxylic acid |
NA |
134896|169824|134896.29 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
(3R,5S)-5-[[(2E)-2-[[5-[3,5-bis(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid |
NA |
134896|169824|134896.29 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
(3R,5S)-5-[[(2E)-2-[[5-[2-chloro-4-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid |
NA |
134896|169824|169824.37 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
(3R,5S)-5-[[(2E)-2-[[5-[2-chloro-5-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid |
NA |
134896|169824|134896.29 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
1-benzyl-N-[(2,4-dichlorophenyl)methyl]piperidin-4-amine |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
2,4-dichloro-N-(1-propylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
2,4-dichloro-N-(1-ethylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
N-(1-benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
N-(1-benzylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
2,4-dichloro-N-piperidin-4-ylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
1-(2-(Tris(4-methoxyphenyl)methoxy)ethyl)piperidine-3-carboxylic acid |
NA |
233000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
2,4-dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A1 |
2-(2-Amino-2-thiazolin-4-yl)acetic acid |
NA |
178000|178800|158489.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A1 |
2,4-dichloro-N-(1-methylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |