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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A1 Nipecotic acid, S-(+)- NA 116000 NA NA NA NA BindingDB|TTD
SLC6A1 (R)-1-(2-(Tris(4-methoxyphenyl)methoxy)ethyl)piperidine-3-carboxylic acid NA 439000 NA NA NA NA BindingDB|TTD
SLC6A1 N-(1-benzylpiperidin-4-yl)-4-fluorobenzamide NA 300000 NA NA NA NA TTD
SLC6A1 (3S)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid NA 809000 NA NA NA NA BindingDB|TTD
SLC6A1 (3R,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid NA 632000 NA NA NA NA BindingDB|TTD
SLC6A1 (3S,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid NA 270000 NA NA NA NA BindingDB|TTD
SLC6A1 (3R)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid NA 270000 NA NA NA NA BindingDB|TTD
SLC6A1 N-(1-benzylpiperidin-4-yl)-2-ethoxybenzamide NA 500000 NA NA NA NA TTD
SLC6A1 1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid NA 268000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[(4-Methoxy-3-trifluoromethyl-phenyl)-phenyl-(3-trifluoromethyl-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 212000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[Tris-(4-fluoro-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 6740000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{3-[Tris-(4-methoxy-phenyl)-methoxy]-propyl}-piperidine-3-carboxylic acid NA 169000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-ethyl}-piperidine-3-carboxylic acid NA 142000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[Tris-(4-methoxy-phenyl)-methylsulfanyl]-ethyl}-piperidine-3-carboxylic acid NA 142000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[(4-Methoxy-phenyl)-diphenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 178000 NA NA NA NA BindingDB|TTD
SLC6A11 N-(1-Benzylpiperidin-4-yl)-2,3-dimethoxybenzamide NA 500000 NA NA NA NA TTD
SLC6A11 N-(1-benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide NA 405000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD