GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC6A1 |
Nipecotic acid, S-(+)- |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
(R)-1-(2-(Tris(4-methoxyphenyl)methoxy)ethyl)piperidine-3-carboxylic acid |
NA |
439000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
N-(1-benzylpiperidin-4-yl)-4-fluorobenzamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
(3S)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
809000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
(3R,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
632000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
(3S,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
(3R)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
N-(1-benzylpiperidin-4-yl)-2-ethoxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid |
NA |
268000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[(4-Methoxy-3-trifluoromethyl-phenyl)-phenyl-(3-trifluoromethyl-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
212000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[Tris-(4-fluoro-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
6740000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{3-[Tris-(4-methoxy-phenyl)-methoxy]-propyl}-piperidine-3-carboxylic acid |
NA |
169000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
142000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[Tris-(4-methoxy-phenyl)-methylsulfanyl]-ethyl}-piperidine-3-carboxylic acid |
NA |
142000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[(4-Methoxy-phenyl)-diphenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
178000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
N-(1-Benzylpiperidin-4-yl)-2,3-dimethoxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
N-(1-benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide |
NA |
405000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |