GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC6A11 |
2,4-dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-(1-prop-2-ynylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
N-(1-benzylpiperidin-4-yl)-2-methylpropanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-(1-propylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-(1-ethylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
N-(1-benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
CI-966 |
NA |
333000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
Guvacine |
NA |
110000|119000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC6A11 |
N-(1-benzylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2,4-dichloro-N-piperidin-4-ylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
Hinokinin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
Nipecotic Acid |
NA |
106000|110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
2,4-dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
2-(2-Amino-2-thiazolin-4-yl)acetic acid |
NA |
150000|150600|125892.54 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
Tiagabine |
NA |
917000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC6A11 |
2,4-dichloro-N-(1-methylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
Nipecotic acid, S-(+)- |
NA |
2320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
N-(1-benzylpiperidin-4-yl)-4-fluorobenzamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |