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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A11 2,4-dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate NA 1000000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-(1-prop-2-ynylpiperidin-4-yl)benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid NA 1000000 NA NA NA NA TTD
SLC6A11 N-(1-benzylpiperidin-4-yl)-2-methylpropanamide NA 1000000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-(1-propylpiperidin-4-yl)benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-(1-ethylpiperidin-4-yl)benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 N-(1-benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide NA 500000 NA NA NA NA TTD
SLC6A11 CI-966 NA 333000 NA NA NA NA BindingDB|TTD
SLC6A11 Guvacine NA 110000|119000 NA NA NA NA BindingDB|PubChem|TTD
SLC6A11 N-(1-benzylpiperidin-4-yl)benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 2,4-dichloro-N-piperidin-4-ylbenzamide NA 1000000 NA NA NA NA TTD
SLC6A11 Hinokinin NA 500000 NA NA NA NA TTD
SLC6A11 Nipecotic Acid NA 106000|110000 NA NA NA NA BindingDB|TTD
SLC6A11 2,4-dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 2-(2-Amino-2-thiazolin-4-yl)acetic acid NA 150000|150600|125892.54 NA NA NA NA BindingDB|TTD
SLC6A11 Tiagabine NA 917000 NA NA NA NA BindingDB|PubChem|TTD
SLC6A11 2,4-dichloro-N-(1-methylpiperidin-4-yl)benzamide NA 1000000 NA NA NA NA TTD
SLC6A11 Nipecotic acid, S-(+)- NA 2320000 NA NA NA NA BindingDB|TTD
SLC6A11 N-(1-benzylpiperidin-4-yl)-4-fluorobenzamide NA 300000 NA NA NA NA TTD