GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC6A11 |
(3S)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
876000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
(3R,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
2043000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
(3S,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
782000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
(3R)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
3233000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
N-(1-benzylpiperidin-4-yl)-2-ethoxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A11 |
N-(4,4-Diphenyl-3-butenyl)nipecotic acid |
NA |
944000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxylic acid |
NA |
1990000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[(3-Fluoro-4-methoxy-phenyl)-(3-fluoro-phenyl)-phenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
198000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A11 |
1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid |
NA |
1080000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[(4-Methoxy-3-trifluoromethyl-phenyl)-phenyl-(3-trifluoromethyl-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
201000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[Tris-(4-fluoro-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
1270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[Bis-(4-fluoro-phenyl)-(4-methoxy-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
151000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[Bis-(4-methoxy-phenyl)-phenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
382000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-[2-(9-Phenyl-9H-xanthen-9-yloxy)-ethyl]-piperidine-3-carboxylic acid |
NA |
920000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[(4-Methoxy-phenyl)-diphenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
655000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[(4-Methoxy-phenyl)-di-p-tolyl-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
Snap-5114 |
NA |
140000|141254 |
NA |
NA |
NA |
NA |
BindingDB |
SLC6A12 |
1-(2-Tritylsulfanyl-ethyl)-piperidine-3-carboxylic acid |
NA |
435000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
Gamma-Aminobutyric Acid |
NA |
165959|181000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
SLC6A12 |
2,4-dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |