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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A11 (3S)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid NA 876000 NA NA NA NA BindingDB|TTD
SLC6A11 (3R,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid NA 2043000 NA NA NA NA BindingDB|TTD
SLC6A11 (3S,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid NA 782000 NA NA NA NA BindingDB|TTD
SLC6A11 (3R)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid NA 3233000 NA NA NA NA BindingDB|TTD
SLC6A11 N-(1-benzylpiperidin-4-yl)-2-ethoxybenzamide NA 500000 NA NA NA NA TTD
SLC6A11 N-(4,4-Diphenyl-3-butenyl)nipecotic acid NA 944000 NA NA NA NA BindingDB|TTD
SLC6A11 1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxylic acid NA 1990000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[(3-Fluoro-4-methoxy-phenyl)-(3-fluoro-phenyl)-phenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 198000 NA NA NA NA BindingDB|TTD
SLC6A11 1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid NA 1080000 NA NA NA NA BindingDB|TTD
SLC6A12 1-{2-[(4-Methoxy-3-trifluoromethyl-phenyl)-phenyl-(3-trifluoromethyl-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 201000 NA NA NA NA BindingDB|TTD
SLC6A12 1-{2-[Tris-(4-fluoro-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 1270000 NA NA NA NA BindingDB|TTD
SLC6A12 1-{2-[Bis-(4-fluoro-phenyl)-(4-methoxy-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 151000 NA NA NA NA BindingDB|TTD
SLC6A12 1-{2-[Bis-(4-methoxy-phenyl)-phenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 382000 NA NA NA NA BindingDB|TTD
SLC6A12 1-[2-(9-Phenyl-9H-xanthen-9-yloxy)-ethyl]-piperidine-3-carboxylic acid NA 920000 NA NA NA NA BindingDB|TTD
SLC6A12 1-{2-[(4-Methoxy-phenyl)-diphenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 655000 NA NA NA NA BindingDB|TTD
SLC6A12 1-{2-[(4-Methoxy-phenyl)-di-p-tolyl-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 109000 NA NA NA NA BindingDB|TTD
SLC6A12 Snap-5114 NA 140000|141254 NA NA NA NA BindingDB
SLC6A12 1-(2-Tritylsulfanyl-ethyl)-piperidine-3-carboxylic acid NA 435000 NA NA NA NA BindingDB|TTD
SLC6A12 Gamma-Aminobutyric Acid NA 165959|181000 NA NA NA NA BindingDB|PubChem
SLC6A12 2,4-dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD