GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC6A12 |
2,4-dichloro-N-(1-methylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A12 |
Nipecotic acid, S-(+)- |
NA |
6410000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
(R)-1-(2-(Tris(4-methoxyphenyl)methoxy)ethyl)piperidine-3-carboxylic acid |
NA |
630000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
(3S)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
335000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
(3R,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
2900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
(3S,8R)-8-benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid |
NA |
809000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
(3R)-8-benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid |
NA |
436000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
N-(1-benzylpiperidin-4-yl)-2-ethoxybenzamide |
NA |
180000|181970 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
N-(4,4-Diphenyl-3-butenyl)nipecotic acid |
NA |
7210000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxylic acid |
NA |
7210000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A12 |
1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid |
NA |
2660000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A13 |
N-(1-benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide |
NA |
479000|501187 |
NA |
NA |
NA |
NA |
BindingDB |
SLC6A13 |
1H-Imidazole-4-acetic acid, 2-amino-4,5-dihydro- |
NA |
125893|132200 |
NA |
NA |
NA |
NA |
BindingDB |
SLC6A13 |
Beta-Alanine |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
SLC6A14 |
alpha-Methyl-DL-tryptophan |
NA |
250000 |
NA |
NA |
NA |
NA |
GtoPDB |
SLC6A15 |
Desloratadine |
NA |
172000 |
NA |
NA |
NA |
NA |
PubChem |
SLC6A15 |
N-(diaminomethylideneamino)benzamide |
376000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC6A15 |
{[4-(N''-carbamimidoylhydrazinecarbonyl)phenyl]formohydrazido}methanimidamide |
173000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC6A15 |
2-(1-Phenylethylidene)hydrazinecarboximidamide |
273000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC6A15 |
N-[(phenylmethylidene)amino]guanidine |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |