| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A2 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A2 |
4-(Benzhydrylsulfanylmethyl)-2-methyl-1,3-thiazole |
NA |
129800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Cubebin |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A2 |
2-(Benzhydrylsulfinylmethyl)-1,3-thiazole |
NA |
420100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-(Benzhydrylsulfinylmethyl)-2-cyclopropyl-1,3-thiazole |
NA |
687200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-(Benzhydrylsulfinylmethyl)-2-chloro-1,3-thiazole |
NA |
108200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-(Benzhydrylsulfinylmethyl)-2-methyl-1,3-thiazole |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
3-(9H-fluoren-9-yl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-ol |
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-[Bis(4-fluorophenyl)methylsulfinylmethyl]thiophene |
NA |
112600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-[[(4-Methylphenyl)-phenylmethyl]sulfinylmethyl]thiophene |
NA |
152500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-(Benzhydrylsulfinylmethyl)-4-methoxy-6-methylpyrimidine |
NA |
227500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
3-(Benzhydrylsulfinylmethyl)-2-bromothiophene |
NA |
144200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-(Benzhydrylsulfinylmethyl)-2-methoxy-2,3-dihydro-1,3,4-thiadiazole |
NA |
145800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-(Benzhydrylsulfinylmethyl)-3-chlorothiophene |
NA |
188100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-(Benzhydrylsulfinylmethyl)-2,6-dimethylpyrimidine |
NA |
767500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(R)-[(R)-(4-fluorophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
230200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(R)-[(S)-(4-bromophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
365100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[Bis(4-methylphenyl)methylsulfinylmethyl]-1,3-thiazole |
NA |
215500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(S)-[(S)-(4-methoxyphenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
195800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(R)-[(R)-(4-methoxyphenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
261000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |