| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A2 |
5-[Bis(4-fluorophenyl)methylsulfinylmethyl]-1,3-thiazole |
NA |
120800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-(Benzhydrylsulfinylmethyl)-2-butyl-1,3-thiazole |
NA |
164400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(S)-[(S)-(4-fluorophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
129300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(S)-[(R)-(4-fluorophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
104300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-(Benzhydrylsulfinylmethyl)-2-thiophen-2-yl-1,3-thiazole |
NA |
110500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-(Benzhydrylsulfinylmethyl)-4,5-dimethyl-1,3-thiazole |
NA |
107300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(S)-[(S)-(4-methylphenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
163700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-[[(S)-[(S)-(4-bromophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
566400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
5-(Benzhydrylsulfinylmethyl)-2-methoxy-1,3-thiazole |
NA |
138800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-[Bis(4-chlorophenyl)methylsulfinylmethyl]-1,3-thiazole |
NA |
107100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
4-[[(4-Bromophenyl)-phenylmethyl]sulfinylmethyl]-1,3-thiazole |
NA |
109100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
N-(bis(4-fluorophenyl)methyl)-8-methyl-8-aza-bicyclo[3.2.1]octan-3-amine |
152000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| SLC6A2 |
6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquinoline |
128900 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Citalopram |
1000000 |
NA |
NA |
NA |
NA |
NA |
GtoPDB|PubChem |
| SLC6A2 |
4-Hydroxy duloxetine beta-D-glucuronide |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A2 |
5-Hydroxy-6-methoxy duloxetine |
920000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A2 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A2 |
Modafinil |
NA |
283600 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| SLC6A2 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A2 |
Sodium 2-methoxy-5-[(1S)-3-(methylamino)-1-(thiophen-2-yl)propoxy]naphthalen-1-yl sulfate |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |