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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A2 5-[(1S)-3-(Methylamino)-1-(thiophen-2-yl)propoxy]naphthalene-1,2-diol 554000 NA NA NA NA NA TTD
SLC6A2 1-Methoxy-5-((S)-3-methylamino-1-thiophen-2-yl-propoxy)-naphthalen-2-ol 235500 NA NA NA NA NA TTD
SLC6A2 Bip-tyr-thr-pro-lys-thr NA 1000000 NA NA NA NA TTD
SLC6A2 Methyl 2-(4-chlorophenyl)cyclopent-1-enecarboxylate 178000|420000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(3-chlorophenyl)cyclopent-1-enecarboxylate 285000|470000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-methoxyphenyl)cyclopent-1-enecarboxylate 550000|1390000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-tert-butylphenyl)cyclopent-1-enecarboxylate 789000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-(trifluoromethoxy)phenyl)cyclopent-1-enecarboxylate 2884000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-acetylphenyl)cyclopent-1-enecarboxylate 240000|646000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(3-aminophenyl)cyclopent-1-enecarboxylate 247000|1318000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-nitrophenyl)cyclopent-1-enecarboxylate 111000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-chlorophenyl)cyclohex-1-enecarboxylate 314000|993000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(3-chlorophenyl)cyclohex-1-enecarboxylate 339000|871000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(biphenyl-4-yl)cyclohex-1-enecarboxylate 215000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-tert-butylphenyl)cyclohex-1-enecarboxylate 1100000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-(trifluoromethoxy)phenyl)cyclohex-1-enecarboxylate 2540000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-phenylcyclohexene-1-carboxylate 2500000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(3-(trifluoromethyl)phenyl)cyclohex-1-enecarboxylate 2110000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-(trifluoromethyl)phenyl)cyclohex-1-enecarboxylate 2020000 NA NA NA NA NA BindingDB|TTD
SLC6A2 Methyl 2-(4-hydroxyphenyl)cyclohex-1-enecarboxylate 499000|675000 NA NA NA NA NA BindingDB|TTD