| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A2 |
XE7RH9J8MC |
5454000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A2 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A2 |
Armodafinil |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| SLC6A3 |
5-((S)-3-Methylamino-1-thiophen-2-yl-propoxy)-naphthalen-2-ol |
163500 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A3 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A3 |
(S)-N-isobutyl-N-(pyrrolidin-3-yl)-2-naphthamide |
NA |
744000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A3 |
US9085531, 4-(3,5-dimethyl-isoxazol-4-yl |
128000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| SLC6A3 |
2-(Benzhydrylsulfinylmethyl)-5-methylpyrimidine |
NA |
155700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A3 |
5-(Benzhydrylsulfinylmethyl)-2-methoxy-2,3-dihydro-1,3,4-thiadiazole |
NA |
107600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A3 |
2-(benzhydrylsulfinylmethyl)-4-methyl-1H-pyrimidin-6-one |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A3 |
4-(Benzhydrylsulfinylmethyl)-2,3-dimethylthiophene |
NA |
283600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A3 |
5-[Bis(4-methylphenyl)methylsulfinylmethyl]-1,3-thiazole |
NA |
356000 |
NA |
NA |
NA |
NA |
BindingDB |
| SLC6A3 |
5-[[(R)-[(S)-(4-methylphenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
133600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A3 |
4-[Bis(4-methoxyphenyl)methylsulfinylmethyl]-2-cyclopropyl-1,3-thiazole |
NA |
104700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A3 |
6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquinoline |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A3 |
Citalopram |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| SLC6A3 |
4-((1S)-3-(Methylamino)-1-(2-thienyl)propoxy)-1-naphthalenol |
130000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A3 |
4-Hydroxy duloxetine beta-D-glucuronide |
3509000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A3 |
5-Hydroxy-6-methoxy duloxetine |
2814000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A3 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |