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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A3 Meropenem NA NA NA NA NA 300000 PubChem
SLC6A3 6-Hydroxy-8-methyl-3-phenyl-8-aza-bicyclo[3.2.1]oct-2-ene-2-carboxylic acid methyl ester NA 150000 NA NA NA NA TTD
SLC6A3 Sodium 2-methoxy-5-[(1S)-3-(methylamino)-1-(thiophen-2-yl)propoxy]naphthalen-1-yl sulfate 10000000 NA NA NA NA NA TTD
SLC6A3 5-[(1S)-3-(Methylamino)-1-(thiophen-2-yl)propoxy]naphthalene-1,2-diol 7275000 NA NA NA NA NA TTD
SLC6A3 1-Methoxy-5-((S)-3-methylamino-1-thiophen-2-yl-propoxy)-naphthalen-2-ol 353000 NA NA NA NA NA TTD
SLC6A3 5-Hydroxyduloxetine 240500 NA NA NA NA NA TTD
SLC6A3 Methyl 2-(4-methoxyphenyl)cyclopent-1-enecarboxylate 140000 NA NA NA NA NA BindingDB
SLC6A3 Methyl 2-(4-tert-butylphenyl)cyclopent-1-enecarboxylate 302000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-(trifluoromethoxy)phenyl)cyclopent-1-enecarboxylate 2649000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-acetylphenyl)cyclopent-1-enecarboxylate 335000 NA NA NA NA NA BindingDB
SLC6A3 Methyl 2-(3-aminophenyl)cyclopent-1-enecarboxylate 121000|875000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(biphenyl-4-yl)cyclohex-1-enecarboxylate 264000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-tert-butylphenyl)cyclohex-1-enecarboxylate 605000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-(trifluoromethoxy)phenyl)cyclohex-1-enecarboxylate 1660000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-phenylcyclohexene-1-carboxylate 630000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(3-(trifluoromethyl)phenyl)cyclohex-1-enecarboxylate 1050000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-(trifluoromethyl)phenyl)cyclohex-1-enecarboxylate 590000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-hydroxyphenyl)cyclohex-1-enecarboxylate 231000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(3-nitrophenyl)cyclohexene-1-carboxylate 239000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(naphthalen-2-yl)cyclohept-1-enecarboxylate 392000 NA NA NA NA NA BindingDB|TTD