GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC6A4 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
SLC6A4 |
Trimethyl-(2-methylsulfonylsulfanylethyl)azanium bromide |
NA |
NA |
NA |
1995262314969 |
NA |
NA |
BindingDB |
SLC6A4 |
1-(4-(Methylsulfonyl)phenyl)propan-2-amine |
NA |
NA |
NA |
2137962.09 |
NA |
NA |
TTD |
SLC6A4 |
Cubebin |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A4 |
4-(Benzhydrylsulfinylmethyl)-2-cyclopropyl-1,3-thiazole |
NA |
436100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
2-[Bis(4-fluorophenyl)methylsulfinylmethyl]thiophene |
NA |
120500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
2-[[(4-Methylphenyl)-phenylmethyl]sulfinylmethyl]thiophene |
NA |
118400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-(Benzhydrylsulfinylmethyl)-3-(trifluoromethyl)-1,2,4-oxadiazole |
NA |
209500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-[[(R)-[(R)-(4-fluorophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
144600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-[Bis(4-methylphenyl)methylsulfinylmethyl]-1,3-thiazole |
NA |
264400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-[[(R)-[(R)-(4-methylphenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
201500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-[[(R)-[(R)-(4-chlorophenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
2-(Benzhydrylsulfinylmethyl)-4,5-dimethyl-1,3-thiazole |
NA |
200800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-[Bis(4-chlorophenyl)methylsulfinylmethyl]-1,3-thiazole |
NA |
220900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
5-[[(S)-[(R)-(4-methoxyphenyl)-phenylmethyl]sulfinyl]methyl]-1,3-thiazole |
NA |
362800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A4 |
4-(1-Methylpyridinium)phenylmethanethiosulphonate iodide |
NA|1300000 |
NA |
NA |
31622776601684|NA |
NA |
NA |
BindingDB |
SLC6A4 |
Tenamfetamine |
NA |
NA |
NA |
1905460|691831 |
NA |
NA |
PubChem |
SLC6A4 |
3,4-Methylenedioxymethamphetamine |
NA |
NA |
NA |
489779 |
NA |
NA |
PubChem |
SLC6A4 |
2-[4-(3-chlorobenzoyl)piperazin-1-yl]-1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]ethanone |
NA |
149000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC6A4 |
1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]-2-[4-(4-methylbenzoyl)piperazin-1-yl]ethanone |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB |