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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A4 2-[4-(3-bromobenzoyl)piperazin-1-yl]-1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]ethanone NA 181000 NA NA NA NA BindingDB
SLC6A4 2-[4-(4-fluorobenzoyl)piperazin-1-yl]-1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]ethanone NA 212000 NA NA NA NA BindingDB
SLC6A4 2-(4-benzoylpiperazin-1-yl)-1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]ethanone NA 320000 NA NA NA NA BindingDB
SLC6A4 2-[4-(4-chlorobenzoyl)piperazin-1-yl]-1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]ethanone NA 546000 NA NA NA NA BindingDB
SLC6A4 1-[4-[3-(5-fluoro-1H-indol-3-yl)propyl]piperazin-1-yl]-2-[4-(4-methoxybenzoyl)piperazin-1-yl]ethanone NA 133000 NA NA NA NA BindingDB
SLC6A4 m-Tolyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate 1000000 NA NA NA NA NA TTD
SLC6A4 4-Hydroxy duloxetine beta-D-glucuronide 10000000 NA NA NA NA NA TTD
SLC6A4 5-Hydroxy-6-methoxy duloxetine 266000 NA NA NA NA NA TTD
SLC6A4 Donepezil NA 1000000 NA NA NA NA PubChem
SLC6A4 4-Methoxyamphetamine NA NA NA 1071520 NA NA PubChem
SLC6A4 Cefazolin NA NA NA NA NA 300000 PubChem
SLC6A4 Modafinil 570000 NA NA NA NA NA BindingDB|PubChem|TTD
SLC6A4 Meropenem NA NA NA NA NA 300000 PubChem
SLC6A4 Hinokinin NA 175000 NA NA NA NA TTD
SLC6A4 Methyl 2-(naphthalen-2-yl)benzoate 620000 NA NA NA NA NA BindingDB
SLC6A4 Sodium 2-methoxy-5-[(1S)-3-(methylamino)-1-(thiophen-2-yl)propoxy]naphthalen-1-yl sulfate 3118000 NA NA NA NA NA TTD
SLC6A4 Methyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate 785000|790000 NA NA NA NA NA BindingDB|TTD
SLC6A4 Methyl 2-(4-chlorophenyl)cyclopent-1-enecarboxylate 2840000 NA NA NA NA NA BindingDB|TTD
SLC6A4 Methyl 2-(3-chlorophenyl)cyclopent-1-enecarboxylate 2240000 NA NA NA NA NA BindingDB|TTD
SLC6A4 Methyl 2-(naphthalen-2-yl)cyclopent-1-enecarboxylate 417000 NA NA NA NA NA BindingDB|TTD