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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC6A3 Methyl 2-(biphenyl-4-yl)cyclohexanecarboxylate 830000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-tert-butylphenyl)cyclohexanecarboxylate 766000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-(trifluoromethoxy)phenyl)cyclohexanecarboxylate 1180000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-phenylcyclohexanecarboxylate 975000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(3-(trifluoromethyl)phenyl)cyclohexanecarboxylate 569000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-(trifluoromethyl)phenyl)cyclohexanecarboxylate 222000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(biphenyl-4-yl)cycloheptanecarboxylate 313000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-tert-butylphenyl)cycloheptanecarboxylate 1140000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 2-(4-tert-butylphenyl)cyclohept-1-enecarboxylate 884000 NA NA NA NA NA BindingDB|TTD
SLC6A3 Methyl 3-(3-nitrophenyl)-7-aza-bicyclo[2.2.1]hept-2-ene-2-carboxylate 232000 NA NA NA NA NA BindingDB|TTD
SLC6A3 H-Asn-Gly-Val-Cys(1)-Cys(2)-Gly-Tyr-Lys-Leu-Cys(2)-His-Hyp-Cys(1)-OH NA 199526.23 NA NA NA NA TTD
SLC6A3 Cefepime NA NA NA NA NA 300000 PubChem
SLC6A3 Ceftazidime NA NA NA NA NA 300000 PubChem
SLC6A3 Aztreonam NA NA NA NA NA 400000 PubChem
SLC6A3 Carumonam NA NA NA NA NA 500000 PubChem
SLC6A3 5-[(1S)-3-(Methylamino)-1-(2-thienyl)propoxy]-1,2-naphthalenediyl bis[I(2)-D-glucopyranosiduronic acid] 10000000 NA NA NA NA NA TTD
SLC6A3 (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-[2-methoxy-5-[(1S)-3-(methylamino)-1-thiophen-2-ylpropoxy]naphthalen-1-yl]oxyoxane-2-carboxylic acid 10000000 NA NA NA NA NA TTD
SLC6A3 XE7RH9J8MC 10000000 NA NA NA NA NA TTD
SLC6A3 Doripenem NA NA NA NA NA 300000 PubChem
SLC6A4 1-(4'-Fluorophenyl)-1-(3-dimethylaminopropyl)-5-bromophthalane NA 120000 NA NA NA NA TTD