| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A4 |
Methyl 2-(3-chlorophenyl)cyclohept-1-enecarboxylate |
463000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(naphthalen-2-yl)cyclohept-1-enecarboxylate |
532000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
1,2-Dichloro-4-(2-(prop-1-enyl)cyclohex-1-enyl)benzene |
381000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(biphenyl-4-yl)cyclohexanecarboxylate |
390000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(4-tert-butylphenyl)cyclohexanecarboxylate |
9120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(4-(trifluoromethoxy)phenyl)cyclohexanecarboxylate |
605000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-phenylcyclohexanecarboxylate |
1510000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(3-(trifluoromethyl)phenyl)cyclohexanecarboxylate |
1910000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(4-(trifluoromethyl)phenyl)cyclohexanecarboxylate |
185000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(4-tert-butylphenyl)cycloheptanecarboxylate |
1800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Methyl 2-(4-tert-butylphenyl)cyclohept-1-enecarboxylate |
1040000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
(2-(3,4-Dichlorophenyl)cyclopent-1-enyl)(morpholino)methanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
(2-(3,4-Dichlorophenyl)cyclopent-1-enyl)(pyrrolidin-1-yl)methanone |
520000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
2-(3,4-dichlorophenyl)-N,N-diethylcyclopent-1-enecarboxamide |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
N-cyclobutyl-2-(3,4-dichlorophenyl)cyclopent-1-enecarboxamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
2-(3,4-dichlorophenyl)-N-(2-fluoroethyl)cyclopent-1-enecarboxamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
2-(3,4-dichlorophenyl)-N-methoxy-N-methylcyclopent-1-enecarboxamide |
540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
2-(3,4-dichlorophenyl)-N-methoxycyclopent-1-enecarboxamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cyclopent-1-enecarboxamide |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Cyclohexyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |