| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A4 |
Isopropyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
2-Fluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
390000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
2,2,2-Trifluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
Phenyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
o-Tolyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
Thiophen-2-ylmethyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
910000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
2-N-Methoxy-N-methylamino-1-(4-methylthiophenyl)propane |
NA |
NA |
NA |
2454708.92 |
NA |
NA |
TTD |
| SLC6A4 |
2-N-(n-Propyl)amino-1-(4-methylthiophenyl)butane |
NA |
NA |
NA |
257039.58 |
NA |
NA |
TTD |
| SLC6A4 |
1-(4-Pentylsulfanylphenyl)propan-1-amine |
NA |
NA |
NA |
1949844.6 |
NA |
NA |
TTD |
| SLC6A4 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A4 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A4 |
5-Dimethylaminobutyryl citalopram |
NA |
NA |
NA |
714000 |
NA |
NA |
BindingDB|TTD |
| SLC6A4 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| SLC6A4 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| SLC6A4 |
Dopamine |
1100000 |
NA |
NA |
NA |
NA |
NA |
PubChem |
| SLC6A4 |
5-[(1S)-3-(Methylamino)-1-(2-thienyl)propoxy]-1,2-naphthalenediyl bis[I(2)-D-glucopyranosiduronic acid] |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
(2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-[2-methoxy-5-[(1S)-3-(methylamino)-1-thiophen-2-ylpropoxy]naphthalen-1-yl]oxyoxane-2-carboxylic acid |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
XE7RH9J8MC |
1459000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A4 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A4 |
Armodafinil |
NA |
232000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |