| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A2 |
Methyl 2-(3-nitrophenyl)cyclohexene-1-carboxylate |
121000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
1,2-Dichloro-4-(2-(prop-1-enyl)cyclohex-1-enyl)benzene |
255000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Methyl 2-(biphenyl-4-yl)cyclohexanecarboxylate |
658000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Methyl 2-(4-tert-butylphenyl)cyclohexanecarboxylate |
675000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Methyl 2-(4-(trifluoromethoxy)phenyl)cyclohexanecarboxylate |
719000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Methyl 2-phenylcyclohexanecarboxylate |
1360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Methyl 2-(3-(trifluoromethyl)phenyl)cyclohexanecarboxylate |
991000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Methyl 2-(4-(trifluoromethyl)phenyl)cyclohexanecarboxylate |
439000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
(2-(3,4-Dichlorophenyl)cyclopent-1-enyl)(morpholino)methanone |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
(2-(3,4-Dichlorophenyl)cyclopent-1-enyl)(pyrrolidin-1-yl)methanone |
410000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-(3,4-dichlorophenyl)-N,N-diethylcyclopent-1-enecarboxamide |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2-(3,4-dichlorophenyl)-N-methoxy-N-methylcyclopent-1-enecarboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Cyclohexyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
2,2,2-Trifluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarboxylate |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A2 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A2 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| SLC6A2 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| SLC6A2 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| SLC6A2 |
5-[(1S)-3-(Methylamino)-1-(2-thienyl)propoxy]-1,2-naphthalenediyl bis[I(2)-D-glucopyranosiduronic acid] |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| SLC6A2 |
(2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-[2-methoxy-5-[(1S)-3-(methylamino)-1-thiophen-2-ylpropoxy]naphthalen-1-yl]oxyoxane-2-carboxylic acid |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |