| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SLC6A12 |
2,4-dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
2,4-dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
2,4-dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
2,4-dichloro-N-(1-prop-2-ynylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
N-(1-benzylpiperidin-4-yl)-2-methylpropanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
2,4-dichloro-N-(1-propylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
2,4-dichloro-N-(1-ethylpiperidin-4-yl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
N-(1-benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide |
NA |
169824|170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A12 |
(-)-Nipecotic acid |
NA |
2310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A12 |
CI-966 |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A12 |
Guvacine |
NA |
1870000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| SLC6A12 |
2,3-Diaminopropionic acid |
NA |
630957 |
NA |
NA |
NA |
NA |
BindingDB |
| SLC6A12 |
N-(1-benzylpiperidin-4-yl)benzamide |
NA |
290000|295121 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A12 |
2,4-dichloro-N-piperidin-4-ylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
Nipecotic Acid |
NA |
2370000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A12 |
1-(2-(Tris(4-methoxyphenyl)methoxy)ethyl)piperidine-3-carboxylic acid |
NA |
140000|208000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SLC6A12 |
2,4-dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SLC6A12 |
Tiagabine |
NA |
1670000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |