GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC5A1 |
3-amino-5-[3-[2,4-dihydroxy-6-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]-3-oxopropyl]-2-hydroxybenzenesulfonic acid |
152000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC5A1 |
4-[5-[3-[2,4-dihydroxy-6-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]-3-oxopropyl]-2-hydroxyanilino]-4-oxobutanoic acid |
116000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC5A11 |
Inositol |
NA |
104000|NA |
NA |
NA|104000 |
NA |
NA |
PubChem |
SLC5A2 |
3,5-diethyl 4-(2H-1,3-benzodioxol-4-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate |
NA |
410930 |
NA |
NA |
NA |
NA |
BindingDB |
SLC5A2 |
(2S,3R,4S,5S,6R)-2-[[5-cyclopropyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol |
NA |
156000 |
NA |
NA |
NA |
NA |
TTD |
SLC5A2 |
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-methoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol |
NA |
204000 |
NA |
NA |
NA |
NA |
TTD |
SLC5A8 |
Ketoprofen |
NA |
119000 |
NA |
NA |
NA |
NA |
GtoPDB |
SLC6A1 |
1-{3-[Tris-(4-methoxy-phenyl)-methoxy]-propyl}-piperidine-3-carboxylic acid |
NA |
121000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
132000|133000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
1-{2-[(4-Methoxy-phenyl)-di-p-tolyl-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
142000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
Snap-5114 |
NA |
170000|388000|389045 |
NA |
NA |
NA |
NA |
BindingDB |
SLC6A1 |
1-{2-[Bis-(4-chloro-phenyl)-(4-methoxy-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC6A1 |
N-(1-Benzylpiperidin-4-yl)-2,3-dimethoxybenzamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
N-(1-benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
2,4-dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
2,4-dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
2,4-dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
(1-Benzylpiperidin-4-yl) 2,4-dichlorobenzoate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
2,4-dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SLC6A1 |
Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |