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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC5A1 3-amino-5-[3-[2,4-dihydroxy-6-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]-3-oxopropyl]-2-hydroxybenzenesulfonic acid 152000 NA NA NA NA NA TTD
SLC5A1 4-[5-[3-[2,4-dihydroxy-6-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]-3-oxopropyl]-2-hydroxyanilino]-4-oxobutanoic acid 116000 NA NA NA NA NA TTD
SLC5A11 Inositol NA 104000|NA NA NA|104000 NA NA PubChem
SLC5A2 3,5-diethyl 4-(2H-1,3-benzodioxol-4-yl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylate NA 410930 NA NA NA NA BindingDB
SLC5A2 (2S,3R,4S,5S,6R)-2-[[5-cyclopropyl-4-[(2-phenylmethoxyphenyl)methyl]-1H-pyrazol-3-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol NA 156000 NA NA NA NA TTD
SLC5A2 (2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-[[4-[(2-methoxyphenyl)methyl]-5-propan-2-yl-1H-pyrazol-3-yl]oxy]oxane-3,4,5-triol NA 204000 NA NA NA NA TTD
SLC5A8 Ketoprofen NA 119000 NA NA NA NA GtoPDB
SLC6A1 1-{3-[Tris-(4-methoxy-phenyl)-methoxy]-propyl}-piperidine-3-carboxylic acid NA 121000 NA NA NA NA BindingDB|TTD
SLC6A1 1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-ethyl}-piperidine-3-carboxylic acid NA 132000|133000 NA NA NA NA BindingDB|TTD
SLC6A1 1-{2-[(4-Methoxy-phenyl)-di-p-tolyl-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 142000 NA NA NA NA BindingDB|TTD
SLC6A1 Snap-5114 NA 170000|388000|389045 NA NA NA NA BindingDB
SLC6A1 1-{2-[Bis-(4-chloro-phenyl)-(4-methoxy-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid NA 122000 NA NA NA NA BindingDB|TTD
SLC6A1 N-(1-Benzylpiperidin-4-yl)-2,3-dimethoxybenzamide NA 500000 NA NA NA NA TTD
SLC6A1 N-(1-benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide NA 1000000 NA NA NA NA TTD
SLC6A1 2,4-dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A1 2,4-dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A1 2,4-dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A1 (1-Benzylpiperidin-4-yl) 2,4-dichlorobenzoate NA 1000000 NA NA NA NA TTD
SLC6A1 2,4-dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide NA 1000000 NA NA NA NA TTD
SLC6A1 Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate NA 1000000 NA NA NA NA TTD