Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
TYR | (2R)-2-amino-3-(1-hydroxy-6-oxopyridin-3-yl)propanoic acid;hydrochloride | NA | 277000 | NA | NA | NA | NA | BindingDB |
TYR | 2,6-Bis(4-hydroxybenzylidene)cyclohexanone | NA | 250000 | NA | NA | NA | NA | TTD |
TYR | Cyclocarposide | NA | 102390 | NA | NA | NA | NA | BindingDB|TTD |
TYR | Benzaldehyde | NA | 820000 | NA | NA | NA | NA | BindingDB|TTD |
TYR | Benzoic Acid | 520000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
TYR | p-Anisaldehyde | NA | 320000 | NA | NA | NA | NA | BindingDB|TTD |
TYR | Kojic acid | NA|350000|730000|1100000 | 125000|133400|280000|400000|500000|571170|2800000|15000000|NA | NA | NA | NA | NA | BindingDB|PubChem |
TYR | Arbutin | NA | 164000|230000|6500000|32000000 | NA | NA | NA | NA | BindingDB|PubChem |
TYR | 1,5-Bis(2-fluoro-4-methoxyphenyl)penta-1,4-dien-3-one | NA | 250000 | NA | NA | NA | NA | TTD |
TYR | 7-Hydroxy-3-(3'',5''-dihydroxyphenyl)coumarin | NA | 10000000 | NA | NA | NA | NA | TTD |
TYR | Resveratrol | NA | 250000|3680000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
TYR | 1-[3-[(1R)-1-[3-acetyl-2,6-dihydroxy-4-methoxy-5-(3-methylbut-2-enyl)phenyl]-3-methylbutyl]-2,4,6-trihydroxy-5-(3-methylbut-2-enyl)phenyl]ethanone | NA | 333000 | NA | NA | NA | NA | BindingDB|TTD |
TYR | Fortuneanoside C | NA | 450000 | NA | NA | NA | NA | BindingDB|TTD |
TYR | 1-hydroxy-5-[(Z)-(4-hydroxy-3-oxo-1-benzofuran-2-ylidene)methyl]pyridin-2-one | NA | 120000 | NA | NA | NA | NA | BindingDB |
TYR | Resorcinol | NA | 3000000 | NA | NA | NA | NA | PubChem |
TYR | Umbelliferone | NA | 420000 | NA | NA | NA | NA | BindingDB|TTD |
TYR | 7-hydroxy-3-phenyl-2H-chromen-2-one | NA | 10000000 | NA | NA | NA | NA | TTD |
TYR | Levodopa | NA | 8400000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
TYR | (1E,4E)-1,5-bis(4-hydroxy-3-methoxyphenyl)penta-1,4-dien-3-one | NA | 250000 | NA | NA | NA | NA | TTD |
TYR | (2S,3R,4S,5S,6R)-2-(2,4-dihydroxyphenoxy)-6-(hydroxymethyl)oxane-3,4,5-triol | NA | 417000 | NA | NA | NA | NA | BindingDB|TTD |