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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
USP7 US10766903, Example 163 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 164 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 165 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 166 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 168 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 169 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 170 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 171 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 173 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 175 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 177 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 199 NA 100500 NA NA NA NA BindingDB
USP7 N-[3-(4-hydroxyphenyl)imidazo[1,2-a]pyridin-2-yl]acetamide NA NA 540000|580000|680000 NA NA NA BindingDB
USP7 4-[(3-Fluorophenoxy)methyl]piperidine NA 2000000 NA NA NA NA TTD
USP7 3H,4H-thieno(2,3-d)pyrimidin-4-one NA NA 471000 NA NA NA BindingDB
USP8 3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one NA 200000 NA NA NA NA TTD
VCAM1 4-Hydroxy-3,3-dimethyl-butyric acid 2,6-di-tert-butyl-4-[1-(3,5-di-tert-butyl-4-hydroxy-phenylsulfanyl)-1-methyl-ethylsulfanyl]-phenyl ester NA 110000 NA NA NA NA BindingDB|TTD
VDR Chenodiol NA NA|150000 NA 150000|NA NA NA PubChem|TTD
VDR H-Leu-Leu-Hse(allyl)(allyl)-Aib-Leu-Leu-Hse(allyl)(allyl)-OH NA 500000 NA NA NA NA BindingDB|TTD
VDR Cholic Acid NA NA|150000 NA 150000|NA NA NA PubChem|TTD