Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
USP7 | US10766903, Example 163 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 164 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 165 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 166 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 168 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 169 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 170 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 171 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 173 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 175 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 177 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 199 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | N-[3-(4-hydroxyphenyl)imidazo[1,2-a]pyridin-2-yl]acetamide | NA | NA | 540000|580000|680000 | NA | NA | NA | BindingDB |
USP7 | 4-[(3-Fluorophenoxy)methyl]piperidine | NA | 2000000 | NA | NA | NA | NA | TTD |
USP7 | 3H,4H-thieno(2,3-d)pyrimidin-4-one | NA | NA | 471000 | NA | NA | NA | BindingDB |
USP8 | 3-acetyl-2-(4-bromophenyl)-1-[2-(3,4-dichlorophenyl)ethyl]-4-hydroxy-2H-pyrrol-5-one | NA | 200000 | NA | NA | NA | NA | TTD |
VCAM1 | 4-Hydroxy-3,3-dimethyl-butyric acid 2,6-di-tert-butyl-4-[1-(3,5-di-tert-butyl-4-hydroxy-phenylsulfanyl)-1-methyl-ethylsulfanyl]-phenyl ester | NA | 110000 | NA | NA | NA | NA | BindingDB|TTD |
VDR | Chenodiol | NA | NA|150000 | NA | 150000|NA | NA | NA | PubChem|TTD |
VDR | H-Leu-Leu-Hse(allyl)(allyl)-Aib-Leu-Leu-Hse(allyl)(allyl)-OH | NA | 500000 | NA | NA | NA | NA | BindingDB|TTD |
VDR | Cholic Acid | NA | NA|150000 | NA | 150000|NA | NA | NA | PubChem|TTD |