GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
XDH |
6-hydroxy-2,4-dioxo-N-(4-(trifluoromethylsulfonamido)phenyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide |
NA |
201000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
2-sulfanylidene-3,6,7,8-tetrahydro-1H-[1,3]thiazino[3,2-a]purin-10-one |
131000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
4-hydroxy-6-oxo-2-sulfanylidene-N-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]-1,3-diazinane-5-carboxamide |
NA |
292000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
2,4,6-trioxo-N-[3-(2H-triazol-4-yl)-1-bicyclo[1.1.1]pentanyl]-1,3-diazinane-5-carboxamide |
NA |
217000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
2-(4-Acetylanilino)-1-[4-(2-aminophenyl)piperazin-1-yl]ethanone |
NA |
20000000000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
2-(4-Acetylanilino)-1-[4-(2-hydroxyphenyl)piperazin-1-yl]ethanone |
NA |
200000000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
Butylated Hydroxyanisole |
NA |
591000 |
NA |
NA |
NA |
NA |
TTD |
XDH |
(3R,4R)-4,8-Dihydroxy-3-((R)-2-Hydroxypentyl)-6,7-Dimethoxyisochroman-1-One |
NA |
612000 |
NA |
NA |
NA |
NA |
TTD |
XDH |
2''-Ethoxy-5''-methoxy-2-(5-methylthienyl)chalcone |
NA |
131000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
8-Bromoxanthine |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
2,6-Diaminopurine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
XDH |
6-Hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
XDH |
Octadecanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester |
NA |
155750 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
Butyric acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester |
NA |
139000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
Acetic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
Tetradecanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
Decanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
Hexanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester |
NA |
129000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
XDH |
Cinnamic Acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB |
XDH |
(-)-6-Feruloyl-catalpol |
NA |
150400 |
NA |
NA |
NA |
NA |
BindingDB|TTD |