Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
XDH 6-hydroxy-2,4-dioxo-N-(4-(trifluoromethylsulfonamido)phenyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide NA 201000 NA NA NA NA BindingDB
XDH 2-sulfanylidene-3,6,7,8-tetrahydro-1H-[1,3]thiazino[3,2-a]purin-10-one 131000 NA NA NA NA NA BindingDB|TTD
XDH 4-hydroxy-6-oxo-2-sulfanylidene-N-[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]-1,3-diazinane-5-carboxamide NA 292000 NA NA NA NA BindingDB
XDH 2,4,6-trioxo-N-[3-(2H-triazol-4-yl)-1-bicyclo[1.1.1]pentanyl]-1,3-diazinane-5-carboxamide NA 217000 NA NA NA NA BindingDB
XDH 2-(4-Acetylanilino)-1-[4-(2-aminophenyl)piperazin-1-yl]ethanone NA 20000000000 NA NA NA NA BindingDB
XDH 2-(4-Acetylanilino)-1-[4-(2-hydroxyphenyl)piperazin-1-yl]ethanone NA 200000000 NA NA NA NA BindingDB
XDH Butylated Hydroxyanisole NA 591000 NA NA NA NA TTD
XDH (3R,4R)-4,8-Dihydroxy-3-((R)-2-Hydroxypentyl)-6,7-Dimethoxyisochroman-1-One NA 612000 NA NA NA NA TTD
XDH 2''-Ethoxy-5''-methoxy-2-(5-methylthienyl)chalcone NA 131000 NA NA NA NA BindingDB|TTD
XDH 8-Bromoxanthine NA 400000 NA NA NA NA BindingDB
XDH 2,6-Diaminopurine NA 200000 NA NA NA NA TTD
XDH 6-Hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid NA 1000000 NA NA NA NA TTD
XDH Octadecanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester NA 155750 NA NA NA NA BindingDB|TTD
XDH Butyric acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester NA 139000 NA NA NA NA BindingDB|TTD
XDH Acetic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester NA 150000 NA NA NA NA BindingDB|TTD
XDH Tetradecanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester NA 102000 NA NA NA NA BindingDB|TTD
XDH Decanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester NA 112000 NA NA NA NA BindingDB|TTD
XDH Hexanoic acid (2S,3R)-2-(3,4-dihydroxy-phenyl)-7,8-dihydroxy-chroman-3-yl ester NA 129000 NA NA NA NA BindingDB|TTD
XDH Cinnamic Acid NA 175000 NA NA NA NA BindingDB
XDH (-)-6-Feruloyl-catalpol NA 150400 NA NA NA NA BindingDB|TTD