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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACR 1-(2-hydroxyethyl)-3-[6-[(3-methoxyphenyl)methylsulfamoyl]-1H-benzimidazol-2-yl]urea NA 7320000 NA NA NA NA BindingDB|TTD
ACR 1-[6-[(3,5-dichlorophenyl)methylsulfamoyl]-1H-benzimidazol-2-yl]-3-(2-hydroxyethyl)urea NA 2450000 NA NA NA NA BindingDB|TTD
ACR 1-[6-[(3,5-difluorophenyl)methylsulfamoyl]-1H-benzimidazol-2-yl]-3-(2-hydroxyethyl)urea NA 340000 NA NA NA NA BindingDB|TTD
ACR 1-(2-hydroxyethyl)-3-[6-[(2-methoxyphenyl)methylsulfamoyl]-1H-benzimidazol-2-yl]urea NA 6040000 NA NA NA NA BindingDB|TTD
ACR 1-(2-hydroxyethyl)-3-[6-[(3-methylphenyl)methylsulfamoyl]-1H-benzimidazol-2-yl]urea NA 5450000 NA NA NA NA BindingDB|TTD
ACR 1-[6-(benzylsulfamoyl)-1H-benzimidazol-2-yl]-3-(2-hydroxyethyl)urea NA 280000 NA NA NA NA BindingDB|TTD
ACR 1-[6-[(2-chlorophenyl)methylsulfamoyl]-1H-benzimidazol-2-yl]-3-(2-hydroxyethyl)urea NA 1060000 NA NA NA NA BindingDB|TTD
ACR 1-[6-(hexylsulfamoyl)-1H-benzimidazol-2-yl]-3-(2-hydroxyethyl)urea NA 1620000 NA NA NA NA BindingDB|TTD
ACR 2-[bis(3-methylbutyl)amino]-N-(6-bromo-1,3-benzothiazol-2-yl)acetamide NA 1090000 NA NA NA NA BindingDB|TTD
ACR N-(6-bromo-1,3-benzothiazol-2-yl)-2-(dipentylamino)acetamide NA 540000 NA NA NA NA BindingDB|TTD
ACR N-(6-bromo-1,3-benzothiazol-2-yl)-2-(4-pentylpiperazin-1-yl)acetamide NA 5080000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxyethyl)-3-(4-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide NA 410000|6810000 NA NA NA NA BindingDB|TTD
ACR N,N-bis(2-hydroxyethyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide NA 5730000 NA NA NA NA BindingDB|TTD
ACR N-(3-hydroxypropyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide NA 1430000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxypropyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide NA 8920000 NA NA NA NA BindingDB|TTD
ACR Ethyl 1-(2,4-dichlorobenzoyl)indazole-3-carboxylate NA 3240000 NA NA NA NA BindingDB|TTD
ACR 1-(2,4-dichlorobenzoyl)-N-methylindazole-3-carboxamide NA 3780000 NA NA NA NA BindingDB|TTD
ACR N-[2-(2-hydroxyethoxy)ethyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide NA 6020000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxyethyl)-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 2700000 NA NA NA NA BindingDB|TTD
ACR N,N-bis(2-hydroxyethyl)-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 5600000 NA NA NA NA BindingDB|TTD