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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACR N-(3-hydroxypropyl)-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 3070000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxypropyl)-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 2950000 NA NA NA NA BindingDB|TTD
ACR N,N-bis(2-hydroxypropyl)-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 1210000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxyethyl)-N-methyl-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 2000000 NA NA NA NA BindingDB|TTD
ACR N-(1-hydroxy-2-methylpropan-2-yl)-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 1875000 NA NA NA NA BindingDB|TTD
ACR N-[2-(2-hydroxyethoxy)ethyl]-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 2070000 NA NA NA NA BindingDB|TTD
ACR N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-3-(4-nitrophenyl)-1H-pyrazole-5-carboxamide NA 5220000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxyethyl)-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 760000 NA NA NA NA BindingDB|TTD
ACR N,N-bis(2-hydroxyethyl)-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 2400000 NA NA NA NA BindingDB|TTD
ACR N-(3-hydroxypropyl)-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 780000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxypropyl)-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 1830000 NA NA NA NA BindingDB|TTD
ACR N-(2-hydroxyethyl)-N-methyl-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 790000 NA NA NA NA BindingDB|TTD
ACR N-[2-(2-hydroxyethoxy)ethyl]-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 9100000 NA NA NA NA BindingDB|TTD
ACR N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-3-(3-nitrophenyl)-1H-pyrazole-5-carboxamide NA 760000 NA NA NA NA BindingDB|TTD
ACR 3-(4-bromophenyl)-N-(2-hydroxyethyl)-1H-pyrazole-5-carboxamide NA 530000 NA NA NA NA BindingDB|TTD
ACR 3-(4-bromophenyl)-N,N-bis(2-hydroxyethyl)-1H-pyrazole-5-carboxamide NA 1520000 NA NA NA NA BindingDB|TTD
ACR 3-(4-bromophenyl)-N-(3-hydroxypropyl)-1H-pyrazole-5-carboxamide NA 380000 NA NA NA NA BindingDB|TTD
ACR 3-(4-bromophenyl)-N-(2-hydroxypropyl)-1H-pyrazole-5-carboxamide NA 330000 NA NA NA NA BindingDB|TTD
ACR 3-(4-bromophenyl)-N-(1-hydroxypropan-2-yl)-1H-pyrazole-5-carboxamide NA 880000 NA NA NA NA BindingDB|TTD
ACR 3-(4-bromophenyl)-N-[2-(2-hydroxyethoxy)ethyl]-1H-pyrazole-5-carboxamide NA 10000000 NA NA NA NA BindingDB|TTD