GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
N-(2-ethylhexyl)-2-thiophenecarboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-[4-(2-methylpiperidin-1-yl)sulfonylphenyl]thiophene-2-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
7-(2-furylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-5,6-diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N,N'-bis(1-methyl-3-phenylpropyl)terephthalamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(4-{5-[1-(2,4-dichlorophenoxy)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)-1,3-benzodioxole-5-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-(3-phenyl-1H-1,2,4-triazol-5-yl)-4-azatricyclo[5.2.1.0~2,6~]dec-8-ene-3,5-dione |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-dione |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
4-{[4-(2-furyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio}-N-(5-methyl-3-isoxazolyl)butanamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(4-methyl-2-oxochromen-7-yl)-2,3-dihydro-1,4-benzodioxine-3-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
3-(4-Chlorophenyl)sulfonyl-2-(furan-2-yl)-1,3-thiazolidine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
ethyl 2,4-dimethyl-5-[2-[[5-(2-phenylpropyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1H-pyrrole-3-carboxylate |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
4-(1-Azabicyclo[2.2.2]oct-2-ylmethyl)benzene-1,2-diol |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
2-Methyl-11-oxo-11H-pyrido(2,1-b)quinazoline-8-carboxylic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
12H-Benzo(g)pyrido(2,1-b)quinazoline-2-carboxylic acid, 12-oxo- |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
2-[1-(1H-benzimidazol-2-yl)-3-(3,5-dimethylphenyl)propan-2-yl]-1H-benzimidazole |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
3-[(2E)-2-(3-methyl-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)quinolin-1(2H)-yl]propane-1-sulfonic acid |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
1-[2-Imino-3-(4-methyl-benzyl)-2,3-dihydro-benzoimidazol-1-yl]-3-phenoxy-propan-2-ol |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
3-Allyl-3a,8a-dihydroxy-1,3,3a,8a-tetrahydro-indeno[1,2-d]imidazole-2,8-dione |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
2-(5-Benzyl-4-phenethyl-4H-[1,2,4]triazol-3-ylsulfanyl)-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
4-amino-N-[2-(cyclopentylamino)-1-(4-methoxyphenyl)-2-oxoethyl]-N-(3-fluorophenyl)-3-(4-fluorophenyl)-1,2-thiazole-5-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |