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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALPG N-(2-ethylhexyl)-2-thiophenecarboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-[4-(2-methylpiperidin-1-yl)sulfonylphenyl]thiophene-2-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 7-(2-furylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-5,6-diphenyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N,N'-bis(1-methyl-3-phenylpropyl)terephthalamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(4-{5-[1-(2,4-dichlorophenoxy)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)-1,3-benzodioxole-5-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 4-(3-phenyl-1H-1,2,4-triazol-5-yl)-4-azatricyclo[5.2.1.0~2,6~]dec-8-ene-3,5-dione NA NA NA 999000 NA NA BindingDB
ALPG 2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-3a,4,7,7a-tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-dione NA NA NA 999000 NA NA BindingDB
ALPG 4-{[4-(2-furyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio}-N-(5-methyl-3-isoxazolyl)butanamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(4-methyl-2-oxochromen-7-yl)-2,3-dihydro-1,4-benzodioxine-3-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 3-(4-Chlorophenyl)sulfonyl-2-(furan-2-yl)-1,3-thiazolidine NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG ethyl 2,4-dimethyl-5-[2-[[5-(2-phenylpropyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]-1H-pyrrole-3-carboxylate NA 999000 NA NA NA NA BindingDB
ALPG 4-(1-Azabicyclo[2.2.2]oct-2-ylmethyl)benzene-1,2-diol NA NA NA 999000 NA NA BindingDB
ALPG 2-Methyl-11-oxo-11H-pyrido(2,1-b)quinazoline-8-carboxylic acid NA 160000 NA NA NA NA BindingDB
ALPG 12H-Benzo(g)pyrido(2,1-b)quinazoline-2-carboxylic acid, 12-oxo- NA 180000 NA NA NA NA BindingDB
ALPG 2-[1-(1H-benzimidazol-2-yl)-3-(3,5-dimethylphenyl)propan-2-yl]-1H-benzimidazole NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 3-[(2E)-2-(3-methyl-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)quinolin-1(2H)-yl]propane-1-sulfonic acid NA NA NA 999000 NA NA BindingDB
ALPG 1-[2-Imino-3-(4-methyl-benzyl)-2,3-dihydro-benzoimidazol-1-yl]-3-phenoxy-propan-2-ol NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 3-Allyl-3a,8a-dihydroxy-1,3,3a,8a-tetrahydro-indeno[1,2-d]imidazole-2,8-dione NA NA NA 999000 NA NA BindingDB
ALPG 2-(5-Benzyl-4-phenethyl-4H-[1,2,4]triazol-3-ylsulfanyl)-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone NA 999000 NA NA NA NA BindingDB
ALPG 4-amino-N-[2-(cyclopentylamino)-1-(4-methoxyphenyl)-2-oxoethyl]-N-(3-fluorophenyl)-3-(4-fluorophenyl)-1,2-thiazole-5-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB