GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
N-[2,5-diethoxy-4-[(2-methylbenzoyl)amino]phenyl]-2H-chromene-3-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-(2-Ethylphenyl)-3-[9-(thiophen-2-ylmethyl)-9-azabicyclo[3.3.1]nonan-3-yl]thiourea |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-[2-(tert-butylamino)-1-(4-fluorophenyl)-2-oxoethyl]-N-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-[5-chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-N'-(6-morpholin-4-ylpyrimidin-4-yl)urea |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
1-(2-Oxo-2-pyrrolidin-1-ylethyl)-3-phenylthieno[3,2-d]pyrimidine-2,4-dione |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
4-[2-{[2-(3,4-dihydroxyphenyl)-2-oxoethyl]thio}-4-oxoquinazolin-3(4H)-yl]-N-(tetrahydrofuran-2-ylmethyl)butanamide |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
5-chloro-N-hexylthiophene-2-sulfonamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
3-methyl-N,6-diphenyl-2-imidazo[2,1-b]thiazolecarboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(4-ethylphenyl)-5-(4-methoxyphenyl)-1,2-oxazole-3-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
5-{[2-(3,4-dihydroxyphenyl)-2-oxoethyl]thio}-2-isopropylimidazo[1,2-c]quinazolin-3(2H)-one |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N-[5-chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-N'-(2-methoxyethyl)urea |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-[5-(Methylamino)-1,3,4-thiadiazol-2-yl]chromen-2-one |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-phenyl-N-[2,2,2-trichloro-1-[(2,5-dimethylphenyl)carbamothioylamino]ethyl]acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-[5-Chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-3-(pyridin-3-ylmethyl)urea |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
[9-(Diphenylphosphoryl)nonyl](diphenyl)phosphine oxide |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
4-Chloro-2-nitro-5-piperidinoaniline |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
(4-Cyanophenyl)methyl 5-oxopyrrolidine-2-carboxylate |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
[2-[(5-Methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl] 2-(4-butan-2-ylphenyl)quinoline-4-carboxylate |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
(4Z)-2-benzyl-4-[[4-(dimethylamino)phenyl]methylidene]-5-methylpyrazol-3-one |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |