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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALPG N-[2,5-diethoxy-4-[(2-methylbenzoyl)amino]phenyl]-2H-chromene-3-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1-(2-Ethylphenyl)-3-[9-(thiophen-2-ylmethyl)-9-azabicyclo[3.3.1]nonan-3-yl]thiourea NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-[2-(tert-butylamino)-1-(4-fluorophenyl)-2-oxoethyl]-N-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-[5-chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-N'-(6-morpholin-4-ylpyrimidin-4-yl)urea NA NA NA 999000 NA NA BindingDB
ALPG 1-(2-Oxo-2-pyrrolidin-1-ylethyl)-3-phenylthieno[3,2-d]pyrimidine-2,4-dione NA 999000 NA NA NA NA BindingDB
ALPG 4-[2-{[2-(3,4-dihydroxyphenyl)-2-oxoethyl]thio}-4-oxoquinazolin-3(4H)-yl]-N-(tetrahydrofuran-2-ylmethyl)butanamide NA NA NA 999000 NA NA BindingDB
ALPG 5-chloro-N-hexylthiophene-2-sulfonamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 3-methyl-N,6-diphenyl-2-imidazo[2,1-b]thiazolecarboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(4-ethylphenyl)-5-(4-methoxyphenyl)-1,2-oxazole-3-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 5-{[2-(3,4-dihydroxyphenyl)-2-oxoethyl]thio}-2-isopropylimidazo[1,2-c]quinazolin-3(2H)-one NA NA NA 999000 NA NA BindingDB
ALPG N-[5-chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-N'-(2-methoxyethyl)urea NA NA NA 999000 NA NA BindingDB
ALPG 3-[5-(Methylamino)-1,3,4-thiadiazol-2-yl]chromen-2-one NA NA NA 999000 NA NA BindingDB
ALPG N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamine NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 2-phenyl-N-[2,2,2-trichloro-1-[(2,5-dimethylphenyl)carbamothioylamino]ethyl]acetamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1-[5-Chloro-2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-3-(pyridin-3-ylmethyl)urea NA NA NA 999000 NA NA BindingDB
ALPG [9-(Diphenylphosphoryl)nonyl](diphenyl)phosphine oxide NA 999000 NA NA NA NA BindingDB
ALPG 4-Chloro-2-nitro-5-piperidinoaniline NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG (4-Cyanophenyl)methyl 5-oxopyrrolidine-2-carboxylate NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG [2-[(5-Methyl-1,2-oxazol-3-yl)amino]-2-oxoethyl] 2-(4-butan-2-ylphenyl)quinoline-4-carboxylate NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG (4Z)-2-benzyl-4-[[4-(dimethylamino)phenyl]methylidene]-5-methylpyrazol-3-one NA NA NA 999000 NA NA BindingDB