GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
1-Butan-2-yl-3-(5-methyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)urea |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-[(3-methoxyphenyl)methyl]-2-[(1-phenyl-5-pyrrol-1-ylpyrazol-4-yl)methylsulfanyl]acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-amino-N'-[(2,4-dichlorobenzyl)oxy]-N-(2-methylphenyl)-1,2,5-oxadiazole-3-carboximidamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
5-(2-Oxo-2-phenylethyl)phenanthridinium |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
Methyl 2-amino-3-(3,4-dihydroxyphenyl)propanoate |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-(4-Chlorophenyl)-5-{[(3-chlorophenyl)sulfanyl]methyl}isoxazole |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
6-Cyclopropyl-2-ethylsulfanyl-4-thiophen-2-ylpyridine-3-carbonitrile |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-ethyl-2,3,4,6-tetrahydro-5H-pyrano[3,2-c]quinolin-5-one |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
3-Hydroxy-3-phenyl-2-[3-(4-sulfamoyl-phenylcarbamoyl)-propionylamino]-propionic acid octyl ester |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-[(1,2-Dimethylindol-5-yl)methyl]-3-(3-methylphenyl)urea |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1'-Butylspiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3'-indole]-2'-one |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(3-methoxyphenyl)-1-[(1-phenyl-5-pyrrol-1-ylpyrazol-4-yl)methyl]piperidine-4-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-[4-(2,4-dimethylphenyl)sulfonylpiperazin-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1''-Allylspiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3''-indoline]-2''-one |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(4-ethylphenyl)-2-[[7-(furan-2-ylmethyl)-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-6-yl]sulfanyl]butanamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-chloro-N-[1-(3,5-dimethylpiperidin-1-yl)-2-methylpropan-2-yl]benzenesulfonamide |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
N-ethyl-3-nitro-N-[(3-nitrophenyl)diazenyl]aniline |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
3-(3,4-Dichlorophenyl)-1-(furan-2-ylmethyl)-1-(1-thiophen-2-ylethyl)urea |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
6-(4-chlorophenyl)-4-(4-methylphenyl)-4,5-dihydro-3(2H)-pyridazinone |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
N-[(1-benzylbenzimidazol-2-yl)methyl]-3-methylaniline |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |