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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALPG 1-Butan-2-yl-3-(5-methyl-6-oxobenzo[b][1,4]benzothiazepin-3-yl)urea NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-[(3-methoxyphenyl)methyl]-2-[(1-phenyl-5-pyrrol-1-ylpyrazol-4-yl)methylsulfanyl]acetamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 4-amino-N'-[(2,4-dichlorobenzyl)oxy]-N-(2-methylphenyl)-1,2,5-oxadiazole-3-carboximidamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 5-(2-Oxo-2-phenylethyl)phenanthridinium NA 999000 NA NA NA NA BindingDB
ALPG Methyl 2-amino-3-(3,4-dihydroxyphenyl)propanoate NA NA NA 999000 NA NA BindingDB
ALPG 3-(4-Chlorophenyl)-5-{[(3-chlorophenyl)sulfanyl]methyl}isoxazole NA 999000 NA NA NA NA BindingDB
ALPG 6-Cyclopropyl-2-ethylsulfanyl-4-thiophen-2-ylpyridine-3-carbonitrile NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 2-ethyl-2,3,4,6-tetrahydro-5H-pyrano[3,2-c]quinolin-5-one NA NA NA 999000 NA NA BindingDB
ALPG 3-Hydroxy-3-phenyl-2-[3-(4-sulfamoyl-phenylcarbamoyl)-propionylamino]-propionic acid octyl ester NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1-[(1,2-Dimethylindol-5-yl)methyl]-3-(3-methylphenyl)urea NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1'-Butylspiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3'-indole]-2'-one NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(3-methoxyphenyl)-1-[(1-phenyl-5-pyrrol-1-ylpyrazol-4-yl)methyl]piperidine-4-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 2-[4-(2,4-dimethylphenyl)sulfonylpiperazin-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1''-Allylspiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3''-indoline]-2''-one NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(4-ethylphenyl)-2-[[7-(furan-2-ylmethyl)-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-6-yl]sulfanyl]butanamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 4-chloro-N-[1-(3,5-dimethylpiperidin-1-yl)-2-methylpropan-2-yl]benzenesulfonamide NA 999000 NA NA NA NA BindingDB
ALPG N-ethyl-3-nitro-N-[(3-nitrophenyl)diazenyl]aniline NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 3-(3,4-Dichlorophenyl)-1-(furan-2-ylmethyl)-1-(1-thiophen-2-ylethyl)urea NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 6-(4-chlorophenyl)-4-(4-methylphenyl)-4,5-dihydro-3(2H)-pyridazinone NA 999000 NA NA NA NA BindingDB
ALPG N-[(1-benzylbenzimidazol-2-yl)methyl]-3-methylaniline NA NA|999000 NA 999000|NA NA NA BindingDB