GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
|
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
2-(2,4-dichlorostyryl)-1H-1,3-benzimidazole |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
|
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
(2,4-Dimethylphenyl)(4-nitrophenyl)methanone |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(5-chloro-2-methoxyphenyl)-2-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]propanamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
(4-Ethoxyphenyl)(1-propyl-1H-benzimidazol-2-yl)methanol |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1,3-Benzodioxol-5-yl(1-propyl-1H-benzimidazol-2-yl)methanol |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
3-(3-phenyl-10H-pyridazino[4,3-b]quinoxalin-5-yl)propan-1-ol |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-(4-Furan-2-ylmethyl-5-phenoxymethyl-4H-[1,2,4]triazol-3-ylsulfanyl)-N-(5-methyl-isoxazol-3-yl)-acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-(1-Adamantyl)-3-[8-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]urea |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
Ethyl 1-[2-(3-fluorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]piperidine-4-carboxylate |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
11-Oxo-11H-pyrido[2,1-b]quinazoline-6-carboxylic acid |
NA |
800000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
1-{1-[4-(Furan-2-carbonyl)-piperazine-1-carbonyl]-cyclohexyl}-3-phenyl-urea |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
5-Methyl-3-(2-propoxy-benzyl)-3H-benzooxazol-2-one |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-[Benzo[1,3]dioxol-5-yl-(2-thiophen-2-yl-acetyl)-amino]-N-cyclohexyl-2-(1-methyl-1H-pyrrol-2-yl)-acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
5-(1,3-benzodioxol-5-yl)-N-(4-chlorobenzyl)-1-methyl-1H-imidazol-2-amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(5-Chloro-2-methoxy-phenyl)-2-[4-(5-methyl-benzotriazol-1-yl)-piperidin-1-yl]-acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-(3,4-Dihydroxy-phenyl)-2-(5-phenyl-4H-[1,2,4]triazol-3-ylsulfanyl)-ethanone |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
5,6-dimethyl-2-[1-[[1-(thiophen-2-ylmethyl)tetrazol-5-yl]methyl]piperidin-4-yl]-1H-benzimidazole |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
5-(4-methoxyphenyl)-N-(pyridin-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |