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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ALPG 5-N,7-dibenzyl-2,6,8,9-tetrahydropyrazolo[3,4-c][2,7]naphthyridine-1,5-diamine NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG Ethyl 1-amino-3-propan-2-yl-3,4-dihydronaphthalene-2-carboxylate NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 14,14-Dimethyl-15-oxa-18-thia-2,9-diazatetracyclo[9.7.0.03,9.012,17]octadeca-1(11),2,12(17)-trien-10-imine;hydrochloride NA NA NA 999000 NA NA BindingDB
ALPG 1-(3-benzyl-2-imino-2,3-dihydro-1H-benzimidazol-1-yl)-3-(4-methoxyphenoxy)propan-2-ol NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(furan-2-ylmethyl)-2-(6-methoxy-2-methyl-4-oxoquinolin-1-yl)acetamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N-(4-ethylphenyl)-3-pyrrol-1-ylthiophene-2-carboxamide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 6-(3-bromophenyl)-3-(3-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine NA NA NA 999000 NA NA BindingDB
ALPG Methyl 2-(5-bromo-4-methoxy-6-methylpyrimidin-2-yl)oxyacetate NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG N,N-dimethyl-4-(1-propan-2-ylbenzimidazol-2-yl)aniline NA 999000 NA NA NA NA BindingDB
ALPG 1-(3,4-Dihydroxyphenyl)-2-[[5-(2-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanone NA NA NA 999000 NA NA BindingDB
ALPG 1-(3,4-Dihydroxyphenyl)-2-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone NA NA NA 999000 NA NA BindingDB
ALPG 2-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1H-benzimidazole NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 5-methyl-N-(3-morpholin-4-ylpropyl)-3-phenylpyrazolo[1,5-a]pyrimidin-7-amine NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 4-Nitrobenzaldehyde N-(4-ethoxybenzyl)thiosemicarbazone NA 999000 NA NA NA NA BindingDB
ALPG 1-benzyl-N'-[(1,3-dimethyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide NA 999000 NA NA NA NA BindingDB
ALPG 1-benzyl-N'-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1-benzyl-N'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 1-benzyl-N'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG 2-[(4-methylbenzyl)sulfanyl]-N'-[(3-methyl-2-thienyl)methylene]acetohydrazide NA NA|999000 NA 999000|NA NA NA BindingDB
ALPG [1-(4-amino-1,2,5-oxadiazol-3-yl)-5-phenyl-1H-1,2,3-triazol-4-yl](phenyl)methanone NA NA|999000 NA 999000|NA NA NA BindingDB