GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ALPG |
5-N,7-dibenzyl-2,6,8,9-tetrahydropyrazolo[3,4-c][2,7]naphthyridine-1,5-diamine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
Ethyl 1-amino-3-propan-2-yl-3,4-dihydronaphthalene-2-carboxylate |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
14,14-Dimethyl-15-oxa-18-thia-2,9-diazatetracyclo[9.7.0.03,9.012,17]octadeca-1(11),2,12(17)-trien-10-imine;hydrochloride |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
1-(3-benzyl-2-imino-2,3-dihydro-1H-benzimidazol-1-yl)-3-(4-methoxyphenoxy)propan-2-ol |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(furan-2-ylmethyl)-2-(6-methoxy-2-methyl-4-oxoquinolin-1-yl)acetamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N-(4-ethylphenyl)-3-pyrrol-1-ylthiophene-2-carboxamide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
6-(3-bromophenyl)-3-(3-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
Methyl 2-(5-bromo-4-methoxy-6-methylpyrimidin-2-yl)oxyacetate |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
N,N-dimethyl-4-(1-propan-2-ylbenzimidazol-2-yl)aniline |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
1-(3,4-Dihydroxyphenyl)-2-[[5-(2-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanone |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
1-(3,4-Dihydroxyphenyl)-2-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethanone |
NA |
NA |
NA |
999000 |
NA |
NA |
BindingDB |
ALPG |
2-[[4-ethyl-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-1H-benzimidazole |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
5-methyl-N-(3-morpholin-4-ylpropyl)-3-phenylpyrazolo[1,5-a]pyrimidin-7-amine |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
4-Nitrobenzaldehyde N-(4-ethoxybenzyl)thiosemicarbazone |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
1-benzyl-N'-[(1,3-dimethyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide |
NA |
999000 |
NA |
NA |
NA |
NA |
BindingDB |
ALPG |
1-benzyl-N'-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-benzyl-N'-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
1-benzyl-N'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methylene]-2,3-dimethyl-1H-indole-5-carbohydrazide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
2-[(4-methylbenzyl)sulfanyl]-N'-[(3-methyl-2-thienyl)methylene]acetohydrazide |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |
ALPG |
[1-(4-amino-1,2,5-oxadiazol-3-yl)-5-phenyl-1H-1,2,3-triazol-4-yl](phenyl)methanone |
NA |
NA|999000 |
NA |
999000|NA |
NA |
NA |
BindingDB |